Compile Data Set for Download or QSAR
Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 9818
TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490791BDBM490791(US10968242, Example 18 | 9-((4S,6R,7S,11aR,13R,14R...)
Affinity DataKi:  0.190nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490777BDBM490777(US10968242, Example 3 Peak 4)
Affinity DataKi:  0.200nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490773BDBM490773(US10968242, Example 2 Peak 4)
Affinity DataKi:  0.200nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490791BDBM490791(US10968242, Example 18 | 9-((4S,6R,7S,11aR,13R,14R...)
Affinity DataKd:  0.200nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490790BDBM490790(US10968242, Example 17 Peak 2)
Affinity DataKd:  0.300nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490790BDBM490790(US10968242, Example 17 Peak 2)
Affinity DataKi:  0.300nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490777BDBM490777(US10968242, Example 3 Peak 4)
Affinity DataKd:  0.300nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490772BDBM490772(US10968242, Example 2 Peak 3)
Affinity DataKd:  0.440nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490790BDBM490790(US10968242, Example 17 Peak 2)
Affinity DataKd:  0.5nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490773BDBM490773(US10968242, Example 2 Peak 4)
Affinity DataKd:  0.780nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490776BDBM490776(US10968242, Example 3 Peak 3)
Affinity DataKi:  1nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490787BDBM490787(US10968242, Example 16 Peak 1)
Affinity DataKi:  1nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490786BDBM490786(US10968242, Example 15 Peak 2)
Affinity DataKi:  1nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490777BDBM490777(US10968242, Example 3 Peak 4)
Affinity DataKd:  1nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490776BDBM490776(US10968242, Example 3 Peak 3)
Affinity DataKd:  1nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490791BDBM490791(US10968242, Example 18 | 9-((4S,6R,7S,11aR,13R,14R...)
Affinity DataKd:  1nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490789BDBM490789(US10968242, Example 17 Peak 1)
Affinity DataKd:  1.5nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490789BDBM490789(US10968242, Example 17 Peak 1)
Affinity DataKi:  2nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490772BDBM490772(US10968242, Example 2 Peak 3)
Affinity DataKi:  2nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490794BDBM490794(US10968242, Example 19 Peak 3)
Affinity DataKd:  2nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490794BDBM490794(US10968242, Example 19 Peak 3)
Affinity DataKi:  2nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490781BDBM490781(US10968242, Example 7 Peak 4)
Affinity DataKd:  3nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490781BDBM490781(US10968242, Example 7 Peak 4)
Affinity DataKd:  3nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490787BDBM490787(US10968242, Example 16 Peak 1)
Affinity DataKd:  3nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490786BDBM490786(US10968242, Example 15 Peak 2)
Affinity DataKd:  3nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490794BDBM490794(US10968242, Example 19 Peak 3)
Affinity DataKd:  3nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490781BDBM490781(US10968242, Example 7 Peak 4)
Affinity DataKi:  3nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490776BDBM490776(US10968242, Example 3 Peak 3)
Affinity DataKd:  3nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490789BDBM490789(US10968242, Example 17 Peak 1)
Affinity DataKd:  4nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490774BDBM490774(US10968242, Example 3 Peak 1)
Affinity DataKi:  4nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490780BDBM490780(US10968242, Example 7 Peak 3)
Affinity DataKd:  4nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490772BDBM490772(US10968242, Example 2 Peak 3)
Affinity DataKd:  6nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490786BDBM490786(US10968242, Example 15 Peak 2)
Affinity DataKd:  6nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490770BDBM490770(US10968242, Example 2 Peak 1)
Affinity DataKi:  7nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490774BDBM490774(US10968242, Example 3 Peak 1)
Affinity DataKd:  8nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490784BDBM490784(US10968242, Example 14 | 9-[(4S,6R,7S,11aR,13R,14R...)
Affinity DataKi:  8nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490799BDBM490799(US10968242, Example 21 Peak 2)
Affinity DataKi:  8nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490788BDBM490788(US10968242, Example 16 Peak 2)
Affinity DataKi:  9nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490780BDBM490780(US10968242, Example 7 Peak 3)
Affinity DataKd:  9nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490795BDBM490795(US10968242, Example 19 Peak 4)
Affinity DataKd:  10nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 490773BDBM490773(US10968242, Example 2 Peak 4)
Affinity DataKd:  11nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490780BDBM490780(US10968242, Example 7 Peak 3)
Affinity DataKi:  13nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490775BDBM490775(US10968242, Example 3 Peak 2)
Affinity DataKd:  14nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490784BDBM490784(US10968242, Example 14 | 9-[(4S,6R,7S,11aR,13R,14R...)
Affinity DataKd:  15nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490799BDBM490799(US10968242, Example 21 Peak 2)
Affinity DataKd:  16nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490775BDBM490775(US10968242, Example 3 Peak 2)
Affinity DataKi:  18nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490795BDBM490795(US10968242, Example 19 Peak 4)
Affinity DataKd:  19nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490788BDBM490788(US10968242, Example 16 Peak 2)
Affinity DataKd:  20nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490792BDBM490792(US10968242, Example 19 Peak 1)
Affinity DataKi:  22nMAssay Description:A radioligand binding assay was developed to determine compound interactions were competitive with a tritium-labeled version of the native STING liga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetStimulator of interferon genes protein(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 490770BDBM490770(US10968242, Example 2 Peak 1)
Affinity DataKd:  23nMAssay Description:Surface plasmon resonance (SPR) STING agonist binding studies were carried out using a Biacore T200 instrument (GE Healthcare) at 4° C. in a 150 mM K...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

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