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Found 471 Enz. Inhib. hit(s) with all data for entry = 9828
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418436(US10457677, Example 4 | US10745399, Example 4 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418557(1-(3-Fluoro-5-methoxy- pyridin-4-yl)-7-methoxy-3- ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418559(1-(1,3-Dimethyl-1H-pyrazol- 4-yl)-7-methoxy-3-meth...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418510(1-(3-Fluoro-5-methoxy- pyridin-2-yl)-7-methoxy-3- ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418561(1-(3-Ethylpyridin-4-yl)-7- methoxy-3-methyl-8-(1- ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418434(US10457677, Example 2 | US10745399, Example 2 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418435(1-[5-(azetidin-3-ylmethoxy)-3-fluoropyridin-2-yl]-...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418436(US10457677, Example 4 | US10745399, Example 4 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418437(US10457677, Example 5 | US10745399, Example 5 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418438(1-[5-(dimethylphosphinoylmethoxy)-3-fluoropyridin-...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418439(US10457677, Example 7 | US10745399, Example 7 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418440(US10457677, Example 8 | US10745399, Example 8 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418441(US10457677, Example 9 | US10745399, Example 9 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418442(US10457677, Example 10 | US10745399, Example 10 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418443(US10457677, Example 11 | US10745399, Example 11 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418444(US10457677, Example 12 | US10745399, Example 12 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418445(US10457677, Example 13 | US10745399, Example 13 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418446(US10457677, Example 14 | US10745399, Example 14 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418447(1-(3-Fluoro-5- methoxypyridin-4-yl)-7- methoxy-3-m...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418448(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoropyrid...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418449(7-Methoxy-3-methyl-1-(1- methyl-1H-pyrazol-4-yl)-8...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418452(1-(3-Fluoro-5-methylpyridin- 2-yl)-7-methoxy-3-met...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418453(1-(1,3-Dimethyl-1H-pyrazol- 4-yl)-8-(1-ethyl-1H-py...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418454(1-(3,5-Difluoropyridin-4-yl)- 7-methoxy-3-methyl-8...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418456(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoropyridin-2-...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418457(1-(3-Ethyl-5-fluoropyridin-4- yl)-8-(1-ethyl-1H-py...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418458(1-(3,5-Difluoropyridin-4-yl)- 8-(1-ethyl-1H-pyrazo...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418459(1-(3-Fluoro-5-methylpyridin- 2-yl)-7-methoxy-3-met...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418465(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoropyridin-4-...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418472(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoro-5-methylp...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418473(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoro-5-me...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418477(7-Methoxy-3-methyl-1-(3- methyl-1H-pyrazol-4-yl)-8...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418566(1-(3-Fluoro-5-methyl- sulfonylmethoxypyridin-2- yl...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418567(1-(3-Cyclopropyl-5-fluoro- pyridin-4-yl)-7-methoxy...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418568(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoro-5-me...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418569(1-(5-Allyloxy-3-fluoropyridin- 2-yl)-7-methoxy-3-m...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418570(1-[5-(Azetidin-3-yloxy)-3- fluoropyridin-2-yl]-7- ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418434(US10457677, Example 2 | US10745399, Example 2 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418435(1-[5-(azetidin-3-ylmethoxy)-3-fluoropyridin-2-yl]-...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418436(US10457677, Example 4 | US10745399, Example 4 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418437(US10457677, Example 5 | US10745399, Example 5 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418438(1-[5-(dimethylphosphinoylmethoxy)-3-fluoropyridin-...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418439(US10457677, Example 7 | US10745399, Example 7 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418440(US10457677, Example 8 | US10745399, Example 8 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418441(US10457677, Example 9 | US10745399, Example 9 | US...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418442(US10457677, Example 10 | US10745399, Example 10 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418443(US10457677, Example 11 | US10745399, Example 11 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418444(US10457677, Example 12 | US10745399, Example 12 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418445(US10457677, Example 13 | US10745399, Example 13 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine-protein kinase ATM(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM418446(US10457677, Example 14 | US10745399, Example 14 | ...)
Affinity DataIC50: <1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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