Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 9851
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493118BDBM493118(US10981916, Example 25 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493117BDBM493117(US10981916, Example 23 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493115BDBM493115(US10981916, Example 21 | 3-cyclopropyl-6-[(5-fluor...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493105BDBM493105(US10981916, Example 19 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493098BDBM493098(US10981916, Example 17 | 3-cyclopropyl-6-[(5-metho...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493094BDBM493094(US10981916, Example 13 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493093BDBM493093(US10981916, Example 12 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493086BDBM493086(US10981916, Example 11 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493069BDBM493069(US10981916, Example 10 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493062BDBM493062(US10981916, Example 9 | 3-cyclopropyl-6-methyl-1-{...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493061BDBM493061(US10981916, Example 8 | 3-cyclopropyl-6-[(5-fluoro...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493060BDBM493060(US10981916, Example 5 | 3-cyclopropyl-6-[(5-methox...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493059BDBM493059(US10981916, Example 2 | 3-cyclopropyl-6-[(5-methox...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493058BDBM493058(US10981916, Example 1 | 3-cyclopropyl-6-[(5-methox...)
Affinity DataIC50: 100nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493155BDBM493155(US10981916, Example 15 | 3-cyclopropyl-6-[(5-fluor...)
Affinity DataIC50: 550nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493145BDBM493145(US10981916, Example 7 | 3-cyclopropyl-6-[(5-fluoro...)
Affinity DataIC50: 550nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493134BDBM493134(US10981916, Example 6 | 3-cyclopropyl-6-[(5-methox...)
Affinity DataIC50: 550nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493122BDBM493122(US10981916, Example 3 | 3-cyclopropyl-6-methyl-1-{...)
Affinity DataIC50: 550nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493297BDBM493297(US10981916, Example 26 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 5.50E+3nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493296BDBM493296(US10981916, Example 24 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 5.50E+3nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493295BDBM493295(US10981916, Example 22 | 3-cyclopropyl-6-[(5-fluor...)
Affinity DataIC50: 5.50E+3nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493294BDBM493294(US10981916, Example 20 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 5.50E+3nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493293BDBM493293(US10981916, Example 14 | 3-cyclopropyl-6-methyl-1-...)
Affinity DataIC50: 5.50E+3nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493299BDBM493299(US10981916, Example 18 | 3-cyclopropyl-6-[(5-metho...)
Affinity DataIC50: 1.00E+4nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent

TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Human)
Dart Neuroscience

US Patent
LigandChemical structure of BindingDB Monomer ID 493298BDBM493298(US10981916, Example 16 | 3-cyclopropyl-6-[(5-fluor...)
Affinity DataIC50: 1.00E+4nMAssay Description:An IMAP TR-FRET-based phosphodiesterase assay was developed using the PDE2A isoform. IMAP technology is based on high-affinity binding of phosphate b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2021
Entry Details
US Patent