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Found 25 Enz. Inhib. hit(s) with all data for entry = 10260
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523849(US11136320, Compound 8)
Affinity DataIC50:  0.420nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523841(US11136320, Compound 4)
Affinity DataIC50:  1.40nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523847(US11136320, Compound 7)
Affinity DataIC50:  1.5nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523839(US11136320, Compound 1)
Affinity DataIC50:  1.5nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523846(US11136320, Compound 64)
Affinity DataIC50:  1.60nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523861(US11136320, Compound 56)
Affinity DataIC50:  1.60nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523844(US11136320, Compound 62)
Affinity DataIC50:  1.70nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523856(US11136320, Compound 75)
Affinity DataIC50:  1.80nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523851(US11136320, Compound 9)
Affinity DataIC50:  2nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523852(US11136320, Compound 72)
Affinity DataIC50:  2nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523843(N-(5-cyano-4-((tetrahydrothiophene-3-yl)amino)pyri...)
Affinity DataIC50:  2nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523848(US11136320, Compound 69)
Affinity DataIC50:  2.10nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523845(US11136320, Compound 6)
Affinity DataIC50:  2.10nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523863(US11136320, Compound 58)
Affinity DataIC50:  2.10nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523840(US11136320, Compound 59)
Affinity DataIC50:  2.10nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523860(US11136320, Compound 83)
Affinity DataIC50:  2.10nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523858(US11136320, Compound 76)
Affinity DataIC50:  2.10nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523853(US11136320, Compound 16)
Affinity DataIC50:  2.20nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523854(US11136320, Compound 73)
Affinity DataIC50:  2.30nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523850(US11136320, Compound 71)
Affinity DataIC50:  2.40nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523857(US11136320, Compound 27)
Affinity DataIC50:  2.40nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM209325(US11136320, Reference Compound | US9266883, 83)
Affinity DataIC50:  2.90nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523842(US11136320, Compound 60)
Affinity DataIC50:  3nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523859(US11136320, Compound 55)
Affinity DataIC50:  3nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Jacobio Pharmaceuticals

US Patent
LigandPNGBDBM523855(US11136320, Compound 20)
Affinity DataIC50:  4.40nMAssay Description:The FGFR4 kinase inhibition of compounds was tested by using mobility shift assay in this experiment, and the rate of FGFR4 kinase inhibition of comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent