Compile Data Set for Download or QSAR
Report error Found 128 Enz. Inhib. hit(s) with all data for entry = 10249
TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522514BDBM522514(US11161850, Example 12)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522543BDBM522543(US11161850, Example 15)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522547BDBM522547(US11161850, Example 16)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522548BDBM522548(US11161850, Example 17)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522549BDBM522549(US11161850, Example 18)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522550BDBM522550(US11161850, Example 19)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522551BDBM522551(US11161850, Example 20)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522552BDBM522552(US11161850, Example 21)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522555BDBM522555(US11161850, Example 22)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522556BDBM522556(US11161850, Example 23 | US11161850, Example 38)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522559BDBM522559(US11161850, Example 24)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522560BDBM522560(US11161850, Example 25)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522561BDBM522561(US11161850, Example 26)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522562BDBM522562(US11161850, Example 27)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522454BDBM522454(US11161850, Example 1)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522459BDBM522459(US11161850, Example 2)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522490BDBM522490(US11161850, Example 3)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522492BDBM522492(US11161850, Example 4)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522504BDBM522504(US11161850, Example 5)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522507BDBM522507(US11161850, Example 7)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522508BDBM522508(US11161850, Example 8)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522511BDBM522511(US11161850, Example 9)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522512BDBM522512(US11161850, Example 10)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522513BDBM522513(US11161850, Example 11)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522671BDBM522671(US11161850, Example 44)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522672BDBM522672(US11161850, Example 45)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522673BDBM522673(US11161850, Example 46)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522674BDBM522674(US11161850, Example 47 | 3-(2-((1H-Indazol-1-yl)me...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522675BDBM522675(US11161850, Example 48 | 3-(2-((1H-Indazol-1-yl)me...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522676BDBM522676(US11161850, Example 49 | US11161850, Example 50 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522676BDBM522676(US11161850, Example 49 | US11161850, Example 50 | ...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522679BDBM522679(US11161850, Example 51 | US11161850, Example 52)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522679BDBM522679(US11161850, Example 51 | US11161850, Example 52)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522681BDBM522681(US11161850, Example 53 | US11161850, Example 54)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522681BDBM522681(US11161850, Example 53 | US11161850, Example 54)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522683BDBM522683(US11161850, Example 55 | US11161850, Example 56)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522683BDBM522683(US11161850, Example 55 | US11161850, Example 56)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522685BDBM522685(US11161850, Example 57 | US11161850, Example 58)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522685BDBM522685(US11161850, Example 57 | US11161850, Example 58)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522687BDBM522687(US11161850, Example 59)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522563BDBM522563(US11161850, Example 28)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522564BDBM522564(US11161850, Example 29 | US11161850, Example 127 |...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522565BDBM522565(US11161850, Example 30)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522566BDBM522566(US11161850, Example 31)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522567BDBM522567(US11161850, Example 32 | 3-(2-((7H-pyrrolo[2,3-b]p...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522568BDBM522568(US11161850, Example 33 | 3-(2-((7H-pyrrolo[2,3-b]p...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522570BDBM522570(US11161850, Example 34)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522571BDBM522571(US11161850, Example 35)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 522572BDBM522572(US11161850, Example 36)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 522573BDBM522573(US11161850, Example 37)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2022
Entry Details
US Patent

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