Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 10325
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528065BDBM528065(US11180482, Example I-46)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528037BDBM528037(US11180482, Example I-18)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528039BDBM528039(US11180482, Example I-20)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528038BDBM528038(US11180482, Example I-19)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528041BDBM528041(US11180482, Example I-22)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528040BDBM528040(US11180482, Example I-21)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528043BDBM528043(US11180482, Example I-24)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 243403BDBM243403(5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(6-me...)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528048BDBM528048(US11180482, Example I-29)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528050BDBM528050(2-((5-chloro-2-((6-methoxy-2-methyl-1,2,3,4-tetrah...)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528020BDBM528020(US11180482, Example I-2)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528024BDBM528024(US11180482, Example I-6)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528057BDBM528057(US11180482, Example I-38)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528023BDBM528023(US11180482, Example I-5)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528059BDBM528059(US11180482, Example I-40)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528058BDBM528058(US11180482, Example I-41 | US11180482, Example I-3...)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528028BDBM528028(US11180482, Example I-10)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528058BDBM528058(US11180482, Example I-41 | US11180482, Example I-3...)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528030BDBM528030(US11180482, Example I-12)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528029BDBM528029(US11180482, Example I-43 | US11180482, Example I-1...)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528029BDBM528029(US11180482, Example I-43 | US11180482, Example I-1...)
Affinity DataIC50: 5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528033BDBM528033(US11180482, Example I-14)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528067BDBM528067(US11180482, Example I-48)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528051BDBM528051(US11180482, Example II-3)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528026BDBM528026(US11180482, Example I-8)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528042BDBM528042(US11180482, Example I-23)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528025BDBM528025(US11180482, Example I-7)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528063BDBM528063(US11180482, Example I-44)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528046BDBM528046(US11180482, Example I-27)
Affinity DataIC50: 7.5nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528031BDBM528031(US11180482, Example I-13)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528036BDBM528036(US11180482, Example I-17)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528019BDBM528019(US11180482, Example I-1)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528022BDBM528022(US11180482, Example I-4)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528055BDBM528055(US11180482, Example I-36)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528021BDBM528021(US11180482, Example I-3)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528056BDBM528056(US11180482, Example I-37)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528045BDBM528045(US11180482, Example I-26)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528061BDBM528061(US11180482, Example I-42)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528027BDBM528027(US11180482, Example I-9)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528047BDBM528047(US11180482, Example I-28)
Affinity DataIC50: 55nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528064BDBM528064(US11180482, Example I-45)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528035BDBM528035(US11180482, Example I-16)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528034BDBM528034(US11180482, Example I-15)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528066BDBM528066(US11180482, Example I-47)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528053BDBM528053(US11180482, Example I-34)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528052BDBM528052(US11180482, Example I-33)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528054BDBM528054(US11180482, Example I-35)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Ariad Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 528044BDBM528044(US11180482, Example I-25)
Affinity DataIC50: 5.05E+3nMAssay Description:The enzymatic activity of Wild Type HPK1 (MAP4K1) Kinase was measured in the presence or absence of an inhibitor compound of the present disclosure b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
US Patent