Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 10353
LigandChemical structure of BindingDB Monomer ID 529895BDBM529895(US11203594, Example 5)
Affinity DataKi:  0.400nMAssay Description:The purpose CDK4/Cyclin D1 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) in the presence of small molecule inhibitors by us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529784BDBM529784(US11203594, Example 2 | WO2020212865, Example 2)
Affinity DataKi:  0.800nMAssay Description:The purpose CDK4/Cyclin D1 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) in the presence of small molecule inhibitors by us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529904BDBM529904(US11203594, Example 15 | US11203594, Example 14)
Affinity DataKi:  0.900nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529893BDBM529893(US11203594, Example 3)
Affinity DataKi:  1.10nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529784BDBM529784(US11203594, Example 2 | WO2020212865, Example 2)
Affinity DataKi:  1.20nMAssay Description:The purpose of the CDK6/Cyclin D3 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) in the presence of small molecule inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529895BDBM529895(US11203594, Example 5)
Affinity DataKi:  1.30nMAssay Description:The purpose of the CDK6/Cyclin D3 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) in the presence of small molecule inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529894BDBM529894(US11203594, Example 4)
Affinity DataKi:  1.60nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529656BDBM529656(US11203594, Example 1)
Affinity DataKi:  1.80nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529919BDBM529919(US11203594, Example 29)
Affinity DataKi:  1.90nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529656BDBM529656(US11203594, Example 1)
Affinity DataKi:  2nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529893BDBM529893(US11203594, Example 3)
Affinity DataKi:  2.10nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529894BDBM529894(US11203594, Example 4)
Affinity DataKi:  2.10nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529902BDBM529902(US11203594, Example 13 | US11203594, Example 12)
Affinity DataKi:  2.10nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529904BDBM529904(US11203594, Example 15 | US11203594, Example 14)
Affinity DataKi:  2.60nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529906BDBM529906(US11203594, Example 17 | US11203594, Example 16)
Affinity DataKi:  2.60nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529898BDBM529898(US11203594, Example 9 | US11203594, Example 8)
Affinity DataKi:  2.70nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529900BDBM529900(US11203594, Example 10)
Affinity DataKi:  2.70nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529912BDBM529912(US11203594, Example 22)
Affinity DataKi:  2.80nMAssay Description:The purpose of the CDK6/Cyclin D3 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) in the presence of small molecule inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529902BDBM529902(US11203594, Example 13 | US11203594, Example 12)
Affinity DataKi:  3.30nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529904BDBM529904(US11203594, Example 15 | US11203594, Example 14)
Affinity DataKi:  3.80nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529909BDBM529909(US11203594, Example 19)
Affinity DataKi:  4.20nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529909BDBM529909(US11203594, Example 19)
Affinity DataKi:  4.5nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529919BDBM529919(US11203594, Example 29)
Affinity DataKi:  4.90nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529906BDBM529906(US11203594, Example 17 | US11203594, Example 16)
Affinity DataKi:  5nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529900BDBM529900(US11203594, Example 10)
Affinity DataKi:  5nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529898BDBM529898(US11203594, Example 9 | US11203594, Example 8)
Affinity DataKi:  6.70nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529896BDBM529896(US11203594, Example 7 | US11203594, Example 6)
Affinity DataKi:  7.20nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529896BDBM529896(US11203594, Example 7 | US11203594, Example 6)
Affinity DataKi:  7.70nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529904BDBM529904(US11203594, Example 15 | US11203594, Example 14)
Affinity DataKi:  7.70nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529902BDBM529902(US11203594, Example 13 | US11203594, Example 12)
Affinity DataKi:  8.5nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529908BDBM529908(US11203594, Example 18)
Affinity DataKi:  9.60nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529902BDBM529902(US11203594, Example 13 | US11203594, Example 12)
Affinity DataKi:  9.70nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529917BDBM529917(US11203594, Example 27)
Affinity DataKi:  9.90nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529918BDBM529918(US11203594, Example 28)
Affinity DataKi:  10nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529906BDBM529906(US11203594, Example 17 | US11203594, Example 16)
Affinity DataKi:  10.5nMAssay Description:The purpose of the CDK6/Cyclin D3 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) in the presence of small molecule inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529914BDBM529914(US11203594, Example 24)
Affinity DataKi:  13nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529916BDBM529916(US11203594, Example 26)
Affinity DataKi:  13nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529911BDBM529911(US11203594, Example 21)
Affinity DataKi:  13nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529911BDBM529911(US11203594, Example 21)
Affinity DataKi:  13nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529922BDBM529922(US11203594, Example 32)
Affinity DataKi:  16nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529901BDBM529901(US11203594, Example 11)
Affinity DataKi:  16nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529914BDBM529914(US11203594, Example 24)
Affinity DataKi:  24nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529917BDBM529917(US11203594, Example 27)
Affinity DataKi:  25nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529921BDBM529921(US11203594, Example 31)
Affinity DataKi:  27nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529922BDBM529922(US11203594, Example 32)
Affinity DataKi:  27nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529921BDBM529921(US11203594, Example 31)
Affinity DataKi:  29nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529908BDBM529908(US11203594, Example 18)
Affinity DataKi:  34nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529901BDBM529901(US11203594, Example 11)
Affinity DataKi:  34nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529915BDBM529915(US11203594, Example 25)
Affinity DataKi:  36nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529918BDBM529918(US11203594, Example 28)
Affinity DataKi:  36nMAssay Description:CDK4/Cyclin D1 and CDK6/Cylcin D3: The Chelation-Enhanced Fluorescence (CHEF) monitors the phosphorylation state in real time where the level of fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2022
Entry Details
US Patent

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