Compile Data Set for Download or QSAR
Report error Found 979 Enz. Inhib. hit(s) with all data for entry = 10409
LigandChemical structure of BindingDB Monomer ID 471418BDBM471418(US10821115, Example 100433 | US11224601, Example 1...)
Affinity DataIC50: 0.0260nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471530BDBM471530(US10821115, Example 100547 | US11224601, Example 1...)
Affinity DataIC50: 0.0310nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 533816BDBM533816(US11224601, Example 271 | (1S,3'R,6'R,7'S,8'E,11'S...)
Affinity DataIC50: 0.0310nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471007BDBM471007(US10821115, Example 100293 | US10821115, Example 1...)
Affinity DataIC50: 0.0320nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471293BDBM471293(US10821115, Example 100308 | US10821115, Example 1...)
Affinity DataIC50: 0.0330nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470885BDBM470885(US10821115, Example 270 | US11224601, Example 270)
Affinity DataIC50: 0.0350nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471363BDBM471363(US10821115, Example 100378 | US11224601, Example 1...)
Affinity DataIC50: 0.0370nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470893BDBM470893(US10821115, Example 278 | (3R)-3-(4- (((1S,3'R,6'R...)
Affinity DataIC50: 0.0390nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471004BDBM471004(US10821115, Example 100327 | US10821115, Example 1...)
Affinity DataIC50: 0.0390nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471430BDBM471430(US10821115, Example 100445 | US11224601, Example 1...)
Affinity DataIC50: 0.0400nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471543BDBM471543(US10821115, Example 100560 | US11224601, Example 1...)
Affinity DataIC50: 0.0410nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471422BDBM471422(US10821115, Example 100437 | US10821115, Example 1...)
Affinity DataIC50: 0.0420nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471416BDBM471416(US10821115, Example 100431 | US11224601, Example 1...)
Affinity DataIC50: 0.0430nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471450BDBM471450(US10821115, Example 100466 | US11224601, Example 1...)
Affinity DataIC50: 0.0430nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471560BDBM471560(US10821115, Example 100577 | US11224601, Example 1...)
Affinity DataIC50: 0.0450nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470777BDBM470777(US10821115, Example 164 | (1S,3'R,6'R,7'S,8'E,10'S...)
Affinity DataIC50: 0.0470nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471292BDBM471292(US10821115, Example 100307 | US11224601, Example 1...)
Affinity DataIC50: 0.0490nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471483BDBM471483(US10821115, Example 100500 | US11224601, Example 1...)
Affinity DataIC50: 0.0490nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471432BDBM471432(US10821115, Example 100447 | US11224601, Example 1...)
Affinity DataIC50: 0.0500nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470833BDBM470833((1S,3''R,6''R,7''R,8''E,11''S,12''R)- 7''-(((9aR)-...)
Affinity DataIC50: 0.0510nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470958BDBM470958(US10821115, Example 341 | (1S,3'R,6'R,7'R,8'E,11'S...)
Affinity DataIC50: 0.0520nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470895BDBM470895(US10821115, Example 280 | (1S,3'R,6'R,7'S,8'E,11'S...)
Affinity DataIC50: 0.0520nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470831BDBM470831(US10821115, Example 215 | US10821115, Example 221 ...)
Affinity DataIC50: 0.0520nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470604BDBM470604((1 S,3′R,6′R,7′R,8′E, 11&#...)
Affinity DataIC50: 0.0530nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471515BDBM471515(US10821115, Example 100532 | US11224601, Example 1...)
Affinity DataIC50: 0.0530nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471420BDBM471420(US10821115, Example 100435 | US10821115, Example 1...)
Affinity DataIC50: 0.0550nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 533926BDBM533926(US11224601, Example 100001 | (1S,3'R,6'R,7'S,8'E, ...)
Affinity DataIC50: 0.0550nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471107BDBM471107(US10821115, Example 100122 | US10821115, Example 1...)
Affinity DataIC50: 0.0560nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471379BDBM471379(US10821115, Example 100394 | US10821115, Example 1...)
Affinity DataIC50: 0.0560nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471408BDBM471408(US10821115, Example 100423 | US11224601, Example 1...)
Affinity DataIC50: 0.0560nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471492BDBM471492(US10821115, Example 100509 | US11224601, Example 1...)
Affinity DataIC50: 0.0570nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 533918BDBM533918(US11224601, Example 405 | (1S,3'R,6'R,7'S,10'S,11'...)
Affinity DataIC50: 0.0570nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471415BDBM471415(US10821115, Example 100430 | US11224601, Example 1...)
Affinity DataIC50: 0.0570nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471528BDBM471528(US10821115, Example 100545 | US10821115, Example 1...)
Affinity DataIC50: 0.0570nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471568BDBM471568(US10821115, Example 100585 | US11224601, Example 1...)
Affinity DataIC50: 0.0570nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470828BDBM470828((1S,3''R,6''R,7''S,8''E,11''S,12''R)- 7''-(((9aS)-...)
Affinity DataIC50: 0.0570nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470849BDBM470849(US10821115, Example 277 | (1S,3''R,6''R,7''S,8''E,...)
Affinity DataIC50: 0.0580nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470603BDBM470603(US10821115, Example 7 | US11224601, Example 7)
Affinity DataIC50: 0.0580nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470816BDBM470816(US10821115, Example 202 | (1S,3'R,6'R,7'S,8'E,11'S...)
Affinity DataIC50: 0.0580nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471533BDBM471533(US10821115, Example 100550 | US11224601, Example 1...)
Affinity DataIC50: 0.0590nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471364BDBM471364(US10821115, Example 100379 | US11224601, Example 1...)
Affinity DataIC50: 0.0600nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470616BDBM470616(US10821115, Example 20 | US11224601, Example 18)
Affinity DataIC50: 0.0600nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470846BDBM470846(US10821115, Example 232 | (1S,3''R,6''R,7''S,8''E,...)
Affinity DataIC50: 0.0610nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470979BDBM470979(US10821115, Example 363 | (1S,3′R,6′R,...)
Affinity DataIC50: 0.0610nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471005BDBM471005(US10821115, Example 100320 | US10821115, Example 1...)
Affinity DataIC50: 0.0610nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470963BDBM470963((1S,3'R,6'R,7'S,8'E,11'S,12'R)- 6-chloro-7'-((9aS)...)
Affinity DataIC50: 0.0620nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471088BDBM471088(US10821115, Example 100101 | US11224601, Example 1...)
Affinity DataIC50: 0.0620nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 470864BDBM470864(US10821115, Example 249 | (1S,3'R,6'R,7'S,8'E,11'S...)
Affinity DataIC50: 0.0630nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471480BDBM471480(US10821115, Example 100497 | US11224601, Example 1...)
Affinity DataIC50: 0.0640nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 471531BDBM471531(US10821115, Example 100548 | US11224601, Example 1...)
Affinity DataIC50: 0.0640nMAssay Description:The inhibition of the Mcl-1/Bim interaction was measured using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The recombinan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2022
Entry Details
US Patent

Displayed 1 to 50 (of 979 total ) | Next | Last >>
Jump to: