Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 10594
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM50260101(CHEMBL4068487 | US10689390, Compound 38 | US113193...)
Affinity DataIC50: <0.5nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448073(US10689390, Compound 23 | US11319326, Compound 23)
Affinity DataIC50:  1nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448074(US10689390, Compound 25 | US11319326, Compound 25)
Affinity DataIC50:  1.60nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM50260078(CHEMBL4095826 | US10689390, Compound 26 | US113193...)
Affinity DataIC50:  2nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM50260080(CHEMBL4088097 | US10689390, Compound 14 | US113193...)
Affinity DataIC50:  3nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448081(US10689390, Compound 37 | US11319326, Compound 37)
Affinity DataIC50:  4nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448083(US10689390, Compound 39 | US11319326, Compound 39)
Affinity DataIC50:  4nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448076(US10689390, Compound 27 | US11319326, Compound 27)
Affinity DataIC50:  4.40nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448078(US10689390, Compound 30 | US11319326, Compound 30)
Affinity DataIC50:  10nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448067(US10689390, Compound 2 | US11319326, Compound 2)
Affinity DataIC50:  10nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM553798(US11319326, Compound 8F)
Affinity DataIC50:  12nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448066(US10689390, Compound 1 | US11319326, Compound 1)
Affinity DataIC50:  24nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448077(US10689390, Compound 28 | US11319326, Compound 28)
Affinity DataIC50:  36nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448079(US10689390, Compound 32 | US11319326, Compound 32)
Affinity DataIC50:  49nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448069(US10689390, Compound 11 | US11319326, Compound 11)
Affinity DataIC50:  61nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448080(US10689390, Compound 35 | US11319326, Compound 35)
Affinity DataIC50:  77nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448071(US10689390, Compound 18 | US11319326, Compound 18)
Affinity DataIC50:  122nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))
Jubilant Biosys

US Patent
LigandPNGBDBM448072(US10689390, Compound 19 | US11319326, Compound 19)
Affinity DataIC50:  176nMAssay Description:Compounds were diluted by step-down dilution method (final concentration of DMSO was 1%) and added to the wells of a 384 well opti plate at desired c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent