Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 10730
LigandChemical structure of BindingDB Monomer ID 562231BDBM562231(US11401274, Example 4 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 2.40nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562247BDBM562247(US11401274, Example 8 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 2.60nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562239BDBM562239(US11401274, Example 7 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 2.70nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562227BDBM562227(US11401274, Example 1 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 2.90nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562228BDBM562228(US11401274, Example 2 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 3nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562227BDBM562227(US11401274, Example 1 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 3.10nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562227BDBM562227(US11401274, Example 1 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 3.30nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562228BDBM562228(US11401274, Example 2 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 4.10nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562235BDBM562235(US11401274, Example 5 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 4.20nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562228BDBM562228(US11401274, Example 2 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 4.30nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562239BDBM562239(US11401274, Example 7 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 5.20nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562236BDBM562236(US11401274, Example 6 | 1-(1-cyclopropylcyclopropy...)
Affinity DataIC50: 5.60nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562235BDBM562235(US11401274, Example 5 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 5.80nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562231BDBM562231(US11401274, Example 4 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 6.30nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562247BDBM562247(US11401274, Example 8 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 6.5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562247BDBM562247(US11401274, Example 8 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 6.60nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562229BDBM562229(US11401274, Example 3 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 6.80nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562231BDBM562231(US11401274, Example 4 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 7.80nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562236BDBM562236(US11401274, Example 6 | 1-(1-cyclopropylcyclopropy...)
Affinity DataIC50: 8.40nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562229BDBM562229(US11401274, Example 3 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 8.70nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562229BDBM562229(US11401274, Example 3 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 9.80nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562239BDBM562239(US11401274, Example 7 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 12nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562236BDBM562236(US11401274, Example 6 | 1-(1-cyclopropylcyclopropy...)
Affinity DataIC50: 14.9nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562229BDBM562229(US11401274, Example 3 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562231BDBM562231(US11401274, Example 4 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562227BDBM562227(US11401274, Example 1 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562228BDBM562228(US11401274, Example 2 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562239BDBM562239(US11401274, Example 7 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562247BDBM562247(US11401274, Example 8 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562235BDBM562235(US11401274, Example 5 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562236BDBM562236(US11401274, Example 6 | 1-(1-cyclopropylcyclopropy...)
Affinity DataIC50: 1.00E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562247BDBM562247(US11401274, Example 8 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.21E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562227BDBM562227(US11401274, Example 1 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.27E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562228BDBM562228(US11401274, Example 2 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.32E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562229BDBM562229(US11401274, Example 3 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.64E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562235BDBM562235(US11401274, Example 5 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.92E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562231BDBM562231(US11401274, Example 4 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 2.18E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562236BDBM562236(US11401274, Example 6 | 1-(1-cyclopropylcyclopropy...)
Affinity DataIC50: 3.92E+4nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562236BDBM562236(US11401274, Example 6 | 1-(1-cyclopropylcyclopropy...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562235BDBM562235(US11401274, Example 5 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562247BDBM562247(US11401274, Example 8 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562239BDBM562239(US11401274, Example 7 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562239BDBM562239(US11401274, Example 7 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562228BDBM562228(US11401274, Example 2 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562227BDBM562227(US11401274, Example 1 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562231BDBM562231(US11401274, Example 4 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 562229BDBM562229(US11401274, Example 3 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 1.00E+5nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562235BDBM562235(US11401274, Example 5 | 1-([1,1′-bi(cyclopro...)
Affinity DataIC50: 0nMAssay Description:All 3′, 5′ cyclic nucleotide phosphodiesterase (PDE) enzyme activities are measured with a radiometric enzyme assay based on SPA detectio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent