Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 10732
LigandChemical structure of BindingDB Monomer ID 562424BDBM562424(US11401279, Example 49)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562425BDBM562425(US11401279, Example 51)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562433BDBM562433(US11401279, Example 66)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562408BDBM562408(US11401279, Example 2)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468549BDBM468549(4-((2-(2,2'- dichloro- 3'-(5- isopropyl-1- methyl-...)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562412BDBM562412(US11401279, Example 7)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468552BDBM468552(4-((2-(2,2′-dichloro-3′-(5-(2-hydroxye...)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562410BDBM562410(US11401279, Example 3)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562416BDBM562416(US11401279, Example 10)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562417BDBM562417(US11401279, Example 11)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562415BDBM562415(US11401279, Example 8)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562420BDBM562420(US11401279, Example 15)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562419BDBM562419(US11401279, Example 12)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468553BDBM468553((S)-4- ((2-(2,2'- dichloro- 3'-(5-(2- hydroxy- pro...)
Affinity DataIC50: 1.60nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562409BDBM562409(US11401279, Example 9)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562422BDBM562422(US11401279, Example 47)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468553BDBM468553((S)-4- ((2-(2,2'- dichloro- 3'-(5-(2- hydroxy- pro...)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562413BDBM562413(US11401279, Example 14)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562421BDBM562421(US11401279, Example 16)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562445BDBM562445(US11401279, Example 183)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562429BDBM562429(US11401279, Example 56)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562432BDBM562432(US11401279, Example 65)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562418BDBM562418(US11401279, Example 13)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468550BDBM468550(4-((2-(2,2'- dichloro- 3'-(5- cyclobutyl-1- methyl...)
Affinity DataIC50: 1.90nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562411BDBM562411(US11401279, Example 4)
Affinity DataIC50: 1.90nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562423BDBM562423(US11401279, Example 48)
Affinity DataIC50: 2nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562428BDBM562428(US11401279, Example 55)
Affinity DataIC50: 2.10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562414BDBM562414(US11401279, Example 5)
Affinity DataIC50: 2.10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562407BDBM562407(US11401279, Example 1)
Affinity DataIC50: 2.20nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562430BDBM562430(US11401279, Example 61)
Affinity DataIC50: 2.20nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 395655BDBM395655(US10308644, Example 265 | (R)-4-(2-(2-(2- chloro-3...)
Affinity DataIC50: 2.30nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 395657BDBM395657(US10308644, Example 267 | (R)-4-((2-(2-chloro-3...)
Affinity DataIC50: 2.30nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468460BDBM468460(US10806785, Example 102 | 4-((2-((2'- chloro-3'-(1...)
Affinity DataIC50: 2.40nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562427BDBM562427(US11401279, Example 53)
Affinity DataIC50: 2.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562431BDBM562431(US11401279, Example 63)
Affinity DataIC50: 2.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562434BDBM562434(US11401279, Example 69)
Affinity DataIC50: 2.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 562426BDBM562426(US11401279, Example 52)
Affinity DataIC50: 2.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468548BDBM468548(4-((2-(2,2′-dichloro-3′-(5-ethyl-1-met...)
Affinity DataIC50: 2.90nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468479BDBM468479(4-((2-((2- chloro-3'-(1,5- dimethyl-4,5,6,7- tetra...)
Affinity DataIC50: 3.40nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468442BDBM468442(US10806785, Example 84 | 4-((2-((2,2′-dichlo...)
Affinity DataIC50: 8.30nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 468551BDBM468551(4-((2-(2,2'- dichloro- 3'-(1- methyl-5- (tetrahydr...)
Affinity DataIC50: 18nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent