Compile Data Set for Download or QSAR
Report error Found 125 Enz. Inhib. hit(s) with all data for entry = 10733
LigandChemical structure of BindingDB Monomer ID 415494BDBM415494(US10428087, Example 39 second peak | US10829502, E...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394320BDBM394320(US9975907, Example 40 | US10428087, Example 40 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394290BDBM394290(US9975907, Example 9 | US10428087, Example 9 | US1...)
Affinity DataIC50: 50nMAssay Description:Assay A1 PI3Kδ: The kinase reaction was conducted in 384-well REMP plate from Thermo Fisher Scientific in a final volume of 40 μL. Inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394293BDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394290BDBM394290(US9975907, Example 9 | US10428087, Example 9 | US1...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 415502BDBM415502(US10428087, Example 43 second peak | US10829502, E...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394289BDBM394289(US9975907, Example 8 | US10428087, Example 8 | US1...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394293BDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394325BDBM394325(US9975907, Example 45 | US10428087, Example 45 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 246889BDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:Assay A1 PI3Kδ: The kinase reaction was conducted in 384-well REMP plate from Thermo Fisher Scientific in a final volume of 40 μL. Inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50004547BDBM50004547(CHEMBL2216863 | US9708333, 28 | US10065963, Compou...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394358BDBM394358(US9975907, Example 78 | US10428087, Example 78 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 246889BDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 246889BDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:Assay A1 PI3Kδ: The kinase reaction was conducted in 384-well REMP plate from Thermo Fisher Scientific in a final volume of 40 μL. Inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394313BDBM394313(US9975907, Example 33 | US10428087, Example 33 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394283BDBM394283(US9975907, Example 2 | US10428087, Example 2 | US1...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394314BDBM394314(US9975907, Example 34 | US10428087, Example 34 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50004547BDBM50004547(CHEMBL2216863 | US9708333, 28 | US10065963, Compou...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394345BDBM394345(US9975907, Example 65 | US10428087, Example 65 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50004547BDBM50004547(CHEMBL2216863 | US9708333, 28 | US10065963, Compou...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394346BDBM394346(US9975907, Example 66 | US10428087, Example 66 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394344BDBM394344(US9975907, Example 64 | US10428087, Example 64 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394347BDBM394347(US9975907, Example 67 | US10428087, Example 67 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394300BDBM394300(US9975907, Example 20 | US10428087, Example 20 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394301BDBM394301(US9975907, Example 21 | US10428087, Example 21 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394353BDBM394353(US9975907, Example 73 | US10428087, Example 73 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 124076BDBM124076(US8754089, 3-(3-fluorophenyl)-6-methyl-2-((1R)-1-(...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394354BDBM394354(US9975907, Example 74 | 2-{1-[(2-Amino-9H-purin-6-...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394294BDBM394294(US9975907, Example 13 | US9975907, Example 23 | US...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394329BDBM394329(US9975907, Example 49 | US10428087, Example 49 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394330BDBM394330(US9975907, Example 50 | US10428087, Example 50 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 246889BDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394334BDBM394334(US9975907, Example 54 | US10428087, Example 54 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394292BDBM394292(US9975907, Example 11 | US10428087, Example 11 | U...)
Affinity DataIC50: 50nMAssay Description:Assay A1 PI3Kδ: The kinase reaction was conducted in 384-well REMP plate from Thermo Fisher Scientific in a final volume of 40 μL. Inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394292BDBM394292(US9975907, Example 11 | US10428087, Example 11 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394332BDBM394332(US9975907, Example 52 | US10428087, Example 52 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394293BDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394337BDBM394337(US9975907, Example 57 | US10428087, Example 57 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394294BDBM394294(US9975907, Example 13 | US9975907, Example 23 | US...)
Affinity DataIC50: 50nMAssay Description:Assay A1 PI3Kδ: The kinase reaction was conducted in 384-well REMP plate from Thermo Fisher Scientific in a final volume of 40 μL. Inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394338BDBM394338(US9975907, Example 58 | US10428087, Example 58 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394293BDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:Assay A1 PI3Kδ: The kinase reaction was conducted in 384-well REMP plate from Thermo Fisher Scientific in a final volume of 40 μL. Inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394294BDBM394294(US9975907, Example 13 | US9975907, Example 23 | US...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394339BDBM394339(US9975907, Example 59 | US10428087, Example 59 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394340BDBM394340(US9975907, Example 60 | US10428087, Example 60 | U...)
Affinity DataIC50: 50nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394286BDBM394286(US9975907, Example 5 | US10428087, Example 5 | US1...)
Affinity DataIC50: 75nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394295BDBM394295(US9975907, Example 14 | US10428087, Example 14 | U...)
Affinity DataIC50: 75nMAssay Description:Assay A1 PI3Kδ: The kinase reaction was conducted in 384-well REMP plate from Thermo Fisher Scientific in a final volume of 40 μL. Inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394285BDBM394285(US9975907, Example 4 | US10428087, Example 4 | US1...)
Affinity DataIC50: 75nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394295BDBM394295(US9975907, Example 14 | US10428087, Example 14 | U...)
Affinity DataIC50: 75nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394318BDBM394318(US9975907, Example 38 | US10428087, Example 38 | U...)
Affinity DataIC50: 75nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 394288BDBM394288(US9975907, Example 7 | US10428087, Example 7 | US1...)
Affinity DataIC50: 75nMAssay Description:PI3Kα, PI3Kβ, PI3Kγ: The kinase reaction was conducted in clear-bottom 96-well plate from Thermo Fisher Scientific in a final volume o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
US Patent

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