Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 10740
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM50318482((-)-menthol | CHEMBL470670 | MENTHOL | US11406649,...)
Affinity DataEC50:  3.80E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562648(1-Di(isopropyl)- phosphinoyl- pentane | US11406649...)
Affinity DataEC50:  5.60E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562695(1-Di(isopropyl)- phosphinoyl- hexane | US11406649,...)
Affinity DataEC50:  2.40E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562697(1-Di(isopropyl)- phosphinoyl- heptane | US11406649...)
Affinity DataEC50:  700nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562698(1-Di(isopropyl)- phosphinoyl- octane | US11406649,...)
Affinity DataEC50:  700nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562746(1-Diispropyl- phosphinoyl- nonane | US11406649, Co...)
Affinity DataEC50:  900nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562753(1-Di(sec-butyl) phosphinoyl- 3-methyl-butane | US1...)
Affinity DataEC50:  4.20E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562748(1-Di(sec-butyl)-phosphinoyl-pentane | US11406649, ...)
Affinity DataEC50:  1.70E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562749(1-Di(sec-butyl)- phosphinoyl- hexane | US11406649,...)
Affinity DataEC50:  800nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562750(1-Di(sec-butyl)- phosphinoyl- heptane | US11406649...)
Affinity DataEC50:  1.10E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562751(1-Di(sec-butyl)- phosphinoyl- octane | US11406649,...)
Affinity DataEC50:  1.30E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562752(1-di(iso-butyl) phosphinoyl- pentane | US11406649,...)
Affinity DataEC50:  2.40E+4nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Individual

US Patent
LigandPNGBDBM562747(1-Di(sec-butyl)- phosphinoyl- butane | US11406649,...)
Affinity DataEC50:  1.45E+4nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent