Compile Data Set for Download or QSAR
Report error Found 574 Enz. Inhib. hit(s) with all data for entry = 10944
TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318725BDBM318725(US9624241, Example 257 | 7-(3,5-dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318724BDBM318724(US9624241, Example 256 | 7-(3,5-dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318724BDBM318724(US9624241, Example 256 | 7-(3,5-dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318727BDBM318727(US9624241, Example 259 | (4S)-7-(3,5-dimethylisoxa...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318729BDBM318729(US9624241, Example 261 | (4S)-7-(3,5-dimethylisoxa...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318728BDBM318728(US9624241, Example 260 | (4S)-7-(3,5-dimethylisoxa...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318731BDBM318731(US9624241, Example 263 | 7-(3,5-dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318730BDBM318730(US9624241, Example 262 | 9-(anilinomethyl)-7-(3,5-...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318717BDBM318717(US9624241, Example 249 | (3R)-1-[(4S)-7-(3,5-dimet...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318717BDBM318717(US9624241, Example 249 | (3R)-1-[(4S)-7-(3,5-dimet...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318716BDBM318716(US9624241, Example 248 | (4S)-7-(3,5-dimethylisoxa...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318716BDBM318716(US9624241, Example 248 | (4S)-7-(3,5-dimethylisoxa...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318719BDBM318719(US9624241, Example 251 | (3R)-N-cyclopropyl-1-[(4S...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318719BDBM318719(US9624241, Example 251 | (3R)-N-cyclopropyl-1-[(4S...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318718BDBM318718(US9624241, Example 250 | (3R)-1-[(4S)-7-(3,5-dimet...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318718BDBM318718(US9624241, Example 250 | (3R)-1-[(4S)-7-(3,5-dimet...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318723BDBM318723(US9624241, Example 255 | 7-(3,5-Dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318723BDBM318723(US9624241, Example 255 | 7-(3,5-Dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318722BDBM318722(US9624241, Example 254 | 7-(3,5-Dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318722BDBM318722(US9624241, Example 254 | 7-(3,5-Dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318740BDBM318740(US9624241, Example 269A | 7-(3,5-dimethylisoxazol-...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318740BDBM318740(US9624241, Example 269A | 7-(3,5-dimethylisoxazol-...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318732BDBM318732(US9624241, Example 264 | 7-(3,5-dimethylisoxazol-4...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 420154BDBM420154(9-chloro-7-(3,5-dimethylisoxazol-4-yl)-4-pyridin-2...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 420153BDBM420153(US10464947, Example 265A | 7-(3,5-dimethylisoxazol...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 420153BDBM420153(US10464947, Example 265A | 7-(3,5-dimethylisoxazol...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 580546BDBM580546(US11498926, Example 267B)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 580546BDBM580546(US11498926, Example 267B)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 580188BDBM580188(US11498926, Example 1A)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 580188BDBM580188(US11498926, Example 1A)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318457BDBM318457(7-(3,5-Dimethylisoxazol-4-yl)-1-methyl-4-phenyl-4,...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318457BDBM318457(7-(3,5-Dimethylisoxazol-4-yl)-1-methyl-4-phenyl-4,...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318459BDBM318459(4-[7-(3,5-Dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-tet...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318459BDBM318459(4-[7-(3,5-Dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-tet...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318458BDBM318458(7-(3,5-Dimethylisoxazol-4-yl)-5-methyl-4-phenyl-4,...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318458BDBM318458(7-(3,5-Dimethylisoxazol-4-yl)-5-methyl-4-phenyl-4,...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318468BDBM318468(7-(3,5-Dimethylisoxazol-4-yl)-4-pyridin-2-yl-4,5-d...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318468BDBM318468(7-(3,5-Dimethylisoxazol-4-yl)-4-pyridin-2-yl-4,5-d...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318471BDBM318471(4-Cyclohexyl-7-(3,5-dimethylisoxazol-4-yl)-4,5-dih...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318471BDBM318471(4-Cyclohexyl-7-(3,5-dimethylisoxazol-4-yl)-4,5-dih...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318468BDBM318468(7-(3,5-Dimethylisoxazol-4-yl)-4-pyridin-2-yl-4,5-d...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318468BDBM318468(7-(3,5-Dimethylisoxazol-4-yl)-4-pyridin-2-yl-4,5-d...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318472BDBM318472(7-(3,5-Dimethylisoxazol-4-yl)-4-(tetrahydrofuran-2...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318473BDBM318473(7-(3,5-Dimethylisoxazol-4-yl)-4-(tetrahydrofuran-2...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318475BDBM318475(2-{2-[7-(3,5-Dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318475BDBM318475(2-{2-[7-(3,5-Dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318474BDBM318474(7-(3,5-Dimethylisoxazol-4-yl)-4-(1,3-thiazol-2-yl)...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318474BDBM318474(7-(3,5-Dimethylisoxazol-4-yl)-4-(1,3-thiazol-2-yl)...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [58-164](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318461BDBM318461(7-(3,5-Dimethylisoxazol-4-yl)-4-(3-methoxyphenyl)-...)
Affinity DataIC50: 100nMAssay Description:Table 11: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetBromodomain-containing protein 4 [353-454](Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 318461BDBM318461(7-(3,5-Dimethylisoxazol-4-yl)-4-(3-methoxyphenyl)-...)
Affinity DataIC50: 100nMAssay Description:Table 12: BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

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