Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 11006
TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585090BDBM585090(US11530180, Compound SU15210-0230-01)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585091BDBM585091(US11530180, Compound SU15210-0238-01)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585088BDBM585088((S)-3-(2-(3-cyano-5 guanidinobenzamido)acetamido)-...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585089BDBM585089(US11530180, Compound SU15210-0206-01)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585094BDBM585094((benzyl (2 S)-2-[[2,6-dichloro-4-(1,1-di oxo-1,4-t...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585092BDBM585092((2S)-2-(2,6-dichloro-4-(1H-indazol-6-yl)benzamido)...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585093BDBM585093((2S)-2-(2,6-dichloro-4-morpholinobenzamido)-3-(2-(...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 584989BDBM584989(US11530180, Compound Table 1.5 | US11530180, Compo...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585011BDBM585011(US11530180, Compound Table 1.3)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585096BDBM585096((S)-2-(2,6-dichloro-4-morpholinobenzamido)-3-(2-(3...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 584980BDBM584980(US11530180, Compound Table 1.1)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585097BDBM585097((S)-2-(2,6-dichloro-4-(1H-indazol-6-yl)benzamido)-...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585045BDBM585045(US11530180, Compound Table 1.9 | US11530180, Compo...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585038BDBM585038(US11530180, Compound Table 1.4)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 584989BDBM584989(US11530180, Compound Table 1.5 | US11530180, Compo...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585079BDBM585079((S)-2-(3,5-dichloro-4′-(methylsulfonyl)biphe...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585080BDBM585080((S)-2-(3,5-dichlorobiphenyl-4-ylcarboxamido)-3-(2-...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585081BDBM585081((2S)-2-(3,5-dichlorobiphenyl-4-yl carboxamido)-3-(...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585087BDBM585087((S)-2-(3,5-dichlorobiphenyl-4-ylcarboxamido)-3-(2-...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585085BDBM585085((S)-2-(3,5-dichlorobiphenyl-4-ylcarboxamido)-3-(2-...)
Affinity DataIC50: 100nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585095BDBM585095((2S)-2-[(2,6-dichloro-4-phenyl-benzoyl)amino]-3-[[...)
Affinity DataIC50: 550nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585082BDBM585082((S)-2-(3,5-dichloro-[1,1′-biphenyl]-4-carbox...)
Affinity DataIC50: 550nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585086BDBM585086((S)-2-(3,5-dichlorobiphenyl-4-ylcarboxamido)-3-(2-...)
Affinity DataIC50: 550nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585084BDBM585084((S,E)-2-(3,5-dichlorobiphenyl-4-ylcarboxamido)-3-(...)
Affinity DataIC50: 550nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585053BDBM585053(US11530180, Compound Table 1.8)
Affinity DataIC50: 1.00E+3nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585045BDBM585045(US11530180, Compound Table 1.9 | US11530180, Compo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585051BDBM585051(US11530180, Compound Table 1.7)
Affinity DataIC50: 1.00E+3nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585083BDBM585083((S)-2-(3,5-dichlorobiphenyl-4-ylcarboxamido)-3-(2-...)
Affinity DataIC50: 5.50E+3nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585065BDBM585065(US11530180, Compound Table 1.11 | US11530180, Comp...)
Affinity DataIC50: 1.00E+4nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585065BDBM585065(US11530180, Compound Table 1.11 | US11530180, Comp...)
Affinity DataIC50: 1.00E+4nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585072BDBM585072(US11530180, Compound Table 1.12)
Affinity DataIC50: 1.00E+4nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585074BDBM585074(US11530180, Compound Table 1.13)
Affinity DataIC50: 1.00E+4nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetIntegrin alpha-5/beta-1(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 585078BDBM585078(US11530180, Compound Table 1.14)
Affinity DataIC50: 5.00E+4nMAssay Description:Evaluation of cell attachment to extracellular matrix proteins was performed as previously described by Yokosaki et al, J. Biol. Chem., 271: (39): 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent