Compile Data Set for Download or QSAR
Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 11056
TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588147BDBM588147(1-[4-[[5-[2-(3- chloroanilino)pyrimidin- 5-yl]-3- ...)
Affinity DataIC50: 5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588172BDBM588172(1-[3-[[6-[2-[2- (trifluoromethoxy) anilino]pyrimid...)
Affinity DataIC50: 5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588164BDBM588164(1-[3-[[6-[2-(3- chloro-4-fluoro- anilino)pyrimidin...)
Affinity DataIC50: 5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588175BDBM588175((E)-1-[4-[[6-[2-(3- chloroanilino)pyrimidin- 5-yl]...)
Affinity DataIC50: 5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588166BDBM588166(1-[3-[[6-[2-[3- (trifluoromethoxy) anilino]pyrimid...)
Affinity DataIC50: 5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588146BDBM588146(1-[3-[[5-[2-[3- (trifluoromethyl)anilino] pyrimidi...)
Affinity DataIC50: 5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588169BDBM588169(1-[3-[[6-[2-[(6- methyl-2- pyridyl)amino] pyrimidi...)
Affinity DataIC50: 5.58nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588168BDBM588168(1-[(3S)-3-[[6-[2-[3- (difluoromethoxy) anilino]pyr...)
Affinity DataIC50: 5.60nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588142BDBM588142(1-[3-[[5-[2-(3- chloroanilino) pyrimidin-5-yl]-3-...)
Affinity DataIC50: 6.01nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588144BDBM588144((S)-1-(3-((5-(2-((3- (difluoromethoxy) phenyl)amin...)
Affinity DataIC50: 6.08nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588173BDBM588173(1-[4-[[6-[2-(3- chlorophenoxy) pyrimidin-5-yl]pyra...)
Affinity DataIC50: 6.11nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588176BDBM588176(1-[4-[[5-[2-(3- chloroanilino)pyrimidin- 5-yl]-3-p...)
Affinity DataIC50: 6.70nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588165BDBM588165(1-[(3S)-3-[[6-[2-[2- (trifluoromethoxy) anilino]py...)
Affinity DataIC50: 6.72nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588161BDBM588161(1-[(2S,3R)-3-[[6- [2-(3- chlorophenoxy) pyrimidin-...)
Affinity DataIC50: 6.88nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588167BDBM588167(1-[4-[[6-[2-[3- (difluoromethoxy) phenoxy]pyrimidi...)
Affinity DataIC50: 6.89nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588124BDBM588124(1-[3-[[5-[2-(3-chloro- 2-fluoro- phenoxy)pyrimidin...)
Affinity DataIC50: 6.89nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588139BDBM588139(1-[3-[[5-[2-(3- chlorophenoxy) pyrimidin-5-yl]-3- ...)
Affinity DataIC50: 6.95nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588153BDBM588153(1-[3-[[6-[2-[3-(difluoromethoxy)phenoxy]pyrimidin-...)
Affinity DataIC50: 8.53nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588149BDBM588149(1-[4-[[5-[2-[[6- (trifluoromethyl)-2- pyridyl]amin...)
Affinity DataIC50: 8.84nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588162BDBM588162(1-[(3S)-3-[[6-[2-[3- (trifluoromethoxy) anilino]py...)
Affinity DataIC50: 9.44nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588160BDBM588160(1-[3-[[6-[2-(3- chlorophenoxy) pyrimidin-5-yl]pyra...)
Affinity DataIC50: 9.49nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588131BDBM588131(1-[3-[[5-[2-(3- chlorophenoxy) pyrimidin-5-yl]-3- ...)
Affinity DataIC50: 9.73nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588128BDBM588128(1-[3-[[5-[2-[3- (difluoromethoxy) phenoxy]pyrimidi...)
Affinity DataIC50: 9.98nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588148BDBM588148(1-[4-[[5-[2-[(6-methyl-2-pyridyl)amino]pyrimidin-5...)
Affinity DataIC50: 16.9nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588158BDBM588158(1-[3-[[6-[2-(3- chlorophenoxy) pyrimidin-5-yl]pyra...)
Affinity DataIC50: 17.7nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588141BDBM588141(1-[3-[[5-[2-(3- ethynylphenoxy) pyrimidin-5-yl]-3-...)
Affinity DataIC50: 17.8nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588138BDBM588138(1-[3-[[5-[2-(3- fluorophenoxy) pyrimidin-5-yl]-3- ...)
Affinity DataIC50: 18.1nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588163BDBM588163(1-[(3S)-3-[[6-[2-(3- chloroanilino) pyrimidin-5-yl...)
Affinity DataIC50: 18.3nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588154BDBM588154(1-[3-[[6-[2-(3- fluorophenoxy) pyrimidin-5-yl]pyra...)
Affinity DataIC50: 19.3nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588171BDBM588171(1-[3-[[6-[2-(3- methoxyphenoxy) pyrimidin-5- yl]py...)
Affinity DataIC50: 19.4nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588132BDBM588132(1-[3-[[5-[2-[3- (trifluoromethyl)phenoxy] pyrimidi...)
Affinity DataIC50: 23.1nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588151BDBM588151((E)-1-[4-[[5-[2-(3-chloroanilino)pyrimidin-5-yl]-3...)
Affinity DataIC50: 24.1nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588123BDBM588123(1-[4-[[5-[2-(3-chlorophenoxy)pyrimidin-5-yl]-3-pyr...)
Affinity DataIC50: 25.3nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588155BDBM588155(1-[3-[[6-[2-[3- (trifluoromethyl) phenoxy]pyrimidi...)
Affinity DataIC50: 30.2nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588150BDBM588150(1-[4-[[5-[2-(2- pyridylamino) pyrimidin-5-yl]-3- p...)
Affinity DataIC50: 31nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588145BDBM588145(1-{(3S)-3-[(5-{2-[(6- methylpyridin-2- yl)amino]py...)
Affinity DataIC50: 32.9nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588156BDBM588156(1-[3-[[6-[2-[3- (trifluoromethoxy) phenoxy]pyrimid...)
Affinity DataIC50: 33.7nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588137BDBM588137(1-[3-[[5-[2-[3- (trifluoromethoxy) phenoxy]pyrimid...)
Affinity DataIC50: 34.5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588164BDBM588164(1-[3-[[6-[2-(3- chloro-4-fluoro- anilino)pyrimidin...)
Affinity DataIC50: 37.3nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588140BDBM588140(1-[3-[[5-[2-(3-chloro- 4-fluoro- phenoxy)pyrimidin...)
Affinity DataIC50: 38.2nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588157BDBM588157(1-[3-[[6-(2- phenoxypyrimidin- 5-yl)pyrazin-2- yl]...)
Affinity DataIC50: 42.9nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588159BDBM588159(1-[3-[[6-[2-(3,5- difluorophenoxy) pyrimidin-5- yl...)
Affinity DataIC50: 43.2nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588174BDBM588174((E)-1-[4-[[6-[2-(3-chlorophenoxy)pyrimidin-5-yl]py...)
Affinity DataIC50: 43.8nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588169BDBM588169(1-[3-[[6-[2-[(6- methyl-2- pyridyl)amino] pyrimidi...)
Affinity DataIC50: 54.9nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588129BDBM588129(1-[(3S)-3-[[5-[2-[3-(difluoromethoxy)phenoxy]pyrim...)
Affinity DataIC50: 55.5nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588136BDBM588136(1-[3-[[5-[2-[3- (difluoromethoxy)-4- fluoro- pheno...)
Affinity DataIC50: 60.6nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588130BDBM588130(1-[(3S)-3-[[5-[2,-(3- chlorophenoxy)pyrimidin- 5-y...)
Affinity DataIC50: 72.4nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588127BDBM588127(3-[5-[5-[(1-prop-2- enoylazetidin-3- yl)amino]-3- ...)
Affinity DataIC50: 75.8nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588170BDBM588170(1-[3-[[6-[2-(4- chlorophenoxy) pyrimidin-5-yl] pyr...)
Affinity DataIC50: 96.8nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 588124BDBM588124(1-[3-[[5-[2-(3-chloro- 2-fluoro- phenoxy)pyrimidin...)
Affinity DataIC50: 121nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREEN Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

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