Compile Data Set for Download or QSAR
Report error Found 195 Enz. Inhib. hit(s) with all data for entry = 11059
LigandChemical structure of BindingDB Monomer ID 588216BDBM588216(1-N'-(4-fluorophenyl)-N-[4-[7- methoxy-6-(2-piperi...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588216BDBM588216(1-N'-(4-fluorophenyl)-N-[4-[7- methoxy-6-(2-piperi...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588215BDBM588215(1-N-[4-[6-[2- (dimethylamino)ethylcarbamoyl]- 7-me...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588215BDBM588215(1-N-[4-[6-[2- (dimethylamino)ethylcarbamoyl]- 7-me...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588217BDBM588217(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(2-morp...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588217BDBM588217(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(2-morp...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588216BDBM588216(1-N'-(4-fluorophenyl)-N-[4-[7- methoxy-6-(2-piperi...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588217BDBM588217(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(2-morp...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588218BDBM588218(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(oxetan...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588218BDBM588218(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(oxetan...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588220BDBM588220(1-N-[4-[6-(azetidine-1- carbonyl)-7-methoxyquinoli...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588219BDBM588219(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [(1-me...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588219BDBM588219(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [(1-me...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588211BDBM588211(methyl 4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cycl...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588211BDBM588211(methyl 4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cycl...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588213BDBM588213(1-N-[4-(6-carbamoyl-7- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588213BDBM588213(1-N-[4-(6-carbamoyl-7- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588212BDBM588212(4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cyclopropan...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588213BDBM588213(1-N-[4-(6-carbamoyl-7- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588214BDBM588214(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (methy...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588214BDBM588214(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (methy...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588214BDBM588214(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (methy...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588221BDBM588221(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyazetidi...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588221BDBM588221(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyazetidi...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588222BDBM588222(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2R)...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588223BDBM588223(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2S)...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588222BDBM588222(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2R)...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588222BDBM588222(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2R)...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588224BDBM588224(1-N-[4-(6-cyano-7- methoxyquinolin-4- yl)oxyphenyl...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588223BDBM588223(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2S)...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588223BDBM588223(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2S)...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588225BDBM588225(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(1,3-ox...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588225BDBM588225(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(1,3-ox...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588225BDBM588225(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(1,3-ox...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588237BDBM588237(1-N'-[3-chloro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588237BDBM588237(1-N'-[3-chloro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588236BDBM588236(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588237BDBM588237(1-N'-[3-chloro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588238BDBM588238(methyl 4-[2-fluoro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588238BDBM588238(methyl 4-[2-fluoro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588238BDBM588238(methyl 4-[2-fluoro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588240BDBM588240(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588240BDBM588240(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588239BDBM588239(4-[2-fluoro-4-[[1-[(4- fluorophenyl)carbamoyl]- cy...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588241BDBM588241(1-N'-[3-fluoro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588241BDBM588241(1-N'-[3-fluoro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588240BDBM588240(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588241BDBM588241(1-N'-[3-fluoro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588232BDBM588232(1-N-[4-[6-carbamoyl-7-(3- morpholin-4- ylpropoxy)q...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 588232BDBM588232(1-N-[4-[6-carbamoyl-7-(3- morpholin-4- ylpropoxy)q...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

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