Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 11105
TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590717BDBM590717(5-({5-[2-(3-aminopropoxy)-4-methoxypyridin-3-yl]-1...)
Affinity DataIC50: 0.100nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590724BDBM590724(US11564920, Example 8)
Affinity DataIC50: 0.100nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590742BDBM590742(US11564920, Example 26)
Affinity DataIC50: 0.140nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590727BDBM590727(US11564920, Example 11)
Affinity DataIC50: 0.180nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590723BDBM590723(US11564920, Example 7)
Affinity DataIC50: 0.210nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590730BDBM590730(US11564920, Example 14)
Affinity DataIC50: 0.220nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590719BDBM590719(US11564920, Example 3)
Affinity DataIC50: 0.220nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590718BDBM590718(US11564920, Example 2)
Affinity DataIC50: 0.220nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590720BDBM590720(US11564920, Example 4)
Affinity DataIC50: 0.230nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590725BDBM590725(US11564920, Example 9)
Affinity DataIC50: 0.240nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590738BDBM590738(US11564920, Example 22)
Affinity DataIC50: 0.240nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590731BDBM590731(US11564920, Example 15)
Affinity DataIC50: 0.260nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590745BDBM590745(US11564920, Example 30)
Affinity DataIC50: 0.260nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590735BDBM590735(US11564920, Example 19)
Affinity DataIC50: 0.260nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590722BDBM590722(US11564920, Example 6)
Affinity DataIC50: 0.270nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590737BDBM590737(US11564920, Example 21)
Affinity DataIC50: 0.290nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590726BDBM590726(US11564920, Example 10)
Affinity DataIC50: 0.300nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590733BDBM590733(US11564920, Example 17)
Affinity DataIC50: 0.300nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590740BDBM590740(US11564920, Example 24)
Affinity DataIC50: 0.300nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590752BDBM590752(US11564920, Example 37)
Affinity DataIC50: 0.320nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590721BDBM590721(US11564920, Example 5)
Affinity DataIC50: 0.330nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590728BDBM590728(US11564920, Example 12)
Affinity DataIC50: 0.340nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590736BDBM590736(US11564920, Example 20)
Affinity DataIC50: 0.340nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590734BDBM590734(US11564920, Example 18)
Affinity DataIC50: 0.510nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50524300BDBM50524300(LY2606368 | Prexasertib | US11564920, Example Prex...)
Affinity DataIC50: 0.540nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590736BDBM590736(US11564920, Example 20)
Affinity DataIC50: 0.600nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590750BDBM590750(US11564920, Example 35)
Affinity DataIC50: 0.620nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590748BDBM590748(US11564920, Example 33)
Affinity DataIC50: 0.690nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590753BDBM590753(US11564920, Example 38)
Affinity DataIC50: 0.700nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590751BDBM590751(US11564920, Example 36)
Affinity DataIC50: 0.730nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590741BDBM590741(US11564920, Example 25)
Affinity DataIC50: 0.740nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590729BDBM590729(US11564920, Example 13)
Affinity DataIC50: 0.740nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590746BDBM590746(US11564920, Example 31)
Affinity DataIC50: 0.75nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590747BDBM590747(US11564920, Example 32)
Affinity DataIC50: 0.760nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590739BDBM590739(US11564920, Example 23)
Affinity DataIC50: 0.790nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590744BDBM590744(US11564920, Example 28)
Affinity DataIC50: 0.800nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590749BDBM590749(US11564920, Example 34)
Affinity DataIC50: 1.82nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590732BDBM590732(US11564920, Example 16)
Affinity DataIC50: 3.04nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590743BDBM590743(US11564920, Example 27)
Affinity DataIC50: 3.46nMAssay Description:IMAP TR-FRET Screening Express Kit (R8160) was obtained from Molecular Devices. CHK1 kinase (02-117, Carna Bio), FAM-labeled CHK1tide (R7185, Molecul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590722BDBM590722(US11564920, Example 6)
Affinity DataIC50: 400nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590721BDBM590721(US11564920, Example 5)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590752BDBM590752(US11564920, Example 37)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590739BDBM590739(US11564920, Example 23)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590753BDBM590753(US11564920, Example 38)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590729BDBM590729(US11564920, Example 13)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590742BDBM590742(US11564920, Example 26)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590732BDBM590732(US11564920, Example 16)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590731BDBM590731(US11564920, Example 15)
Affinity DataIC50: 2.70E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590738BDBM590738(US11564920, Example 22)
Affinity DataIC50: 3.00E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 590728BDBM590728(US11564920, Example 12)
Affinity DataIC50: 3.10E+3nMAssay Description:The test compounds were added to cultured hERG (human Ether-a-go-go Related Gene) gene stably expressing CHO cell line cells to achieve 0.27 to 100 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

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