Compile Data Set for Download or QSAR
Report error Found 275 Enz. Inhib. hit(s) with all data for entry = 11176
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597684BDBM597684(US11603377, Compound 5)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 36609BDBM36609(Rapamycin C-7, analog 4 | SIROLIMUS | US11603377, ...)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597683BDBM597683(US11603377, Compound 4)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597715BDBM597715(US11603377, Compound 36)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597686BDBM597686(US11603377, Compound 7)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597685BDBM597685(US11603377, Compound 6)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597688BDBM597688(US11603377, Compound 9)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597687BDBM597687(US11603377, Compound 8)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597708BDBM597708(US11603377, Compound 35 | US11603377, Compound 29)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597707BDBM597707(US11603377, Compound 34 | US11603377, Compound 28)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597740BDBM597740(US11603377, Compound 61)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597710BDBM597710(US11603377, Compound 31)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597709BDBM597709(US11603377, Compound 30)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597712BDBM597712(US11603377, Compound 33)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597711BDBM597711(US11603377, Compound 32)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597744BDBM597744(US11603377, Compound 65)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597708BDBM597708(US11603377, Compound 35 | US11603377, Compound 29)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597747BDBM597747(US11603377, Compound 68)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597681BDBM597681(US11603377, Compound 2)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597707BDBM597707(US11603377, Compound 34 | US11603377, Compound 28)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597746BDBM597746(US11603377, Compound 67)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597700BDBM597700(US11603377, Compound 21)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597699BDBM597699(US11603377, Compound 20)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597702BDBM597702(US11603377, Compound 23)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597734BDBM597734(US11603377, Compound 55)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597701BDBM597701(US11603377, Compound 22)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597704BDBM597704(US11603377, Compound 25)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597703BDBM597703(US11603377, Compound 24)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597735BDBM597735(US11603377, Compound 56)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597706BDBM597706(US11603377, Compound 27)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597705BDBM597705(US11603377, Compound 26)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597738BDBM597738(US11603377, Compound 59)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597692BDBM597692(US11603377, Compound 16 | US11603377, Compound 13)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597694BDBM597694(US11603377, Compound 15)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597696BDBM597696(US11603377, Compound 17)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597728BDBM597728(US11603377, Compound 49)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597692BDBM597692(US11603377, Compound 16 | US11603377, Compound 13)
Affinity DataKd: <0.300nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597732BDBM597732(US11603377, Compound 53)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597731BDBM597731(US11603377, Compound 52)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597748BDBM597748(US11603377, Compound 69)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597718BDBM597718(US11603377, Compound 39)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597717BDBM597717(US11603377, Compound 38)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597720BDBM597720(US11603377, Compound 41)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597690BDBM597690(US11603377, Compound 11)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597689BDBM597689(US11603377, Compound 10)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597737BDBM597737(US11603377, Compound 58)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597691BDBM597691(US11603377, Compound 12)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597743BDBM597743(US11603377, Compound 64)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597693BDBM597693(US11603377, Compound 14)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Aeovian Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 597745BDBM597745(US11603377, Compound 66)
Affinity DataKd:  0.650nMAssay Description:Biotinylated avi-FKBP12 was immobilized on a streptavidin chip (Cytiva Series S SA) using a Biacore 8K or 8 k+ (Cytiva). To achieve an immobilization...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2023
Entry Details
US Patent

Displayed 1 to 50 (of 275 total ) | Next | Last >>
Jump to: