Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 11195
LigandChemical structure of BindingDB Monomer ID 598702BDBM598702(US11613536, Example 1 | (2S)-1-[(2-{[(2-methylbiph...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598706BDBM598706(US11613536, Example 5 | 5-{[(2-hydroxyethyl)amino]...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598703BDBM598703(US11613536, Example 2 | 5-{[(2-hydroxyethyl)amino]...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598710BDBM598710(US11613536, Example 9 | 5-{[(2-hydroxyethyl)amino]...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598709BDBM598709(US11613536, Example 8 | 4-chloro-5-{[(2-hydroxyeth...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598708BDBM598708(US11613536, Example 7 | 5-{[(2-hydroxyethyl)amino]...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598707BDBM598707(US11613536, Example 6 | (2S)-1-[(1-methyl-3-{[(2-m...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598714BDBM598714(US11613536, Example 13 | N-[2-cyano-3-(1-methyl-1H...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598713BDBM598713(US11613536, Example 12 | N-(2-cyano-2′-fluor...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598712BDBM598712(US11613536, Example 11 | N-(2-cyano-2′-fluor...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598711BDBM598711(US11613536, Example 10 | N-[2-cyano-3-(2,3-dihydro...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598718BDBM598718(US11613536, Example 17 | (S)-1-(5-chloro-2-((5-cya...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598716BDBM598716(US11613536, Example 15 | N-(2-cyano-2′-fluor...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598715BDBM598715(US11613536, Example 14 | N-[2-cyano-3-(2,3-dihydro...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598720BDBM598720(US11613536, Example 19 | 5-(((R)-3-hydroxypyrrolid...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598719BDBM598719(US11613536, Example 18 | (S)-1-(5-chloro-2-((5-cya...)
Affinity DataIC50: 100nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598717BDBM598717(US11613536, Example 16 | N-[2-cyano-3-(1-methyl-1H...)
Affinity DataIC50: 300nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598705BDBM598705(US11613536, Example 4 | (2S)-1-[(1-methyl-2-{[(2-m...)
Affinity DataIC50: 300nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 598704BDBM598704(US11613536, Example 3 | 5-{[(2-hydroxyethyl)amino]...)
Affinity DataIC50: 300nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2023
Entry Details
US Patent