Compile Data Set for Download or QSAR
Report error Found 472 Enz. Inhib. hit(s) with all data for entry = 11219
TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601106BDBM601106(US11634396, Compound 65 | 2-fluoro-4-((S)-3-((R)-3...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601109BDBM601109(US11634396, Compound 68 | 4-((S)-2-(dimethylamino)...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601211BDBM601211(US11634396, Compound 152 | 4-((S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601108BDBM601108(US11634396, Compound 67 | 4-((S)-3-((S)-3-cyclopro...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601194BDBM601194(US11634396, Compound 150 | 2-chloro-4-((S)-3-((S)-...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601111BDBM601111(US11634396, Compound 70 | 4-[(2S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601212BDBM601212(US11634396, Compound 154 | 4-((S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601218BDBM601218(US11634396, Compound 157 | 4-((S)-3-((S)-4,4-dimet...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601090BDBM601090(4-[(2S)-2-(dimethylamino)-3-[3-(pyridin-3-yl)-3-[1...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601286BDBM601286((S)-N-((S)-3-(1H-indazol-5-yl)-2-(piperidin-1-yl)p...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601089BDBM601089(4-[(2S)-2-(dimethylamino)-3-[3-(6-methoxypyridin-3...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601182BDBM601182(US11634396, Compound 140 | 4-((S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601384BDBM601384((3R)-N-[(2S)-3-[2-chloro-4-(1H-pyrazol-4-yl)phenyl...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601187BDBM601187(US11634396, Compound 143 | 4-((S)-2-(dimethylamino...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601095BDBM601095(4-((S)-2-(dimethylamino)-3-((S)-3-(thiophen-3-yl)-...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601186BDBM601186(US11634396, Compound 142 | 4-((S)-3-((R)-3-(4-chlo...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601189BDBM601189(US11634396, Compound 145 | 4-((S)-2-(dimethylamino...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601099BDBM601099(US11634396, Compound 58 | 4-((S)-2-(dimethylamino)...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601188BDBM601188(US11634396, Compound 144 | 4-((S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601102BDBM601102(US11634396, Compound 61 | 4-((S)-2-(dimethylamino)...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601190BDBM601190(US11634396, Compound 146 | 4-((S)-3-((R)-4,4-dimet...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetKappa-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601290BDBM601290((3R)-N-[(2S)-2-(dimethylamino)-3-(1H-indazol-1-yl)...)
Affinity DataIC50: 300nMAssay Description:KOR β-Arrestin Agonist and Antagonist assays were preformed using the Tango OPRK1-bla U2OS cells from Invitrogen and purchased from ThermoFisher...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 600945BDBM600945(US11634396, Compound 8 | 4-((S)-2-(dimethylamino)-...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601230BDBM601230(US11634396, Compound 167 | 4-((S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601321BDBM601321((R)-N-((S)-3-(2-chloro-3-fluoro-4-methoxyphenyl)-2...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601123BDBM601123(US11634396, Compound 82 | 4-((S)-2-(methylamino)-3...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 600924BDBM600924(US11634396, Compound 7 | 4-((S)-2-(dimethylamino)-...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 600961BDBM600961(US11634396, Compound 9 | 4-[(2S)-2-(dimethylamino)...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601232BDBM601232(US11634396, Compound 169 | (R)-N-((S)-2-(dimethyla...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601231BDBM601231(US11634396, Compound 168 | (S)-3-(((S)-4,4-dimethy...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 600945BDBM600945(US11634396, Compound 8 | 4-((S)-2-(dimethylamino)-...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 600978BDBM600978(US11634396, Compound 10 | 4-((S)-2-(dimethylamino)...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601234BDBM601234((3S)-N-[(2S)-2-(dimethylamino)-3-(7-methyl-2-oxo-2...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601051BDBM601051(4-[(2S)-2-(dimethylamino)-3-[(3R)-5-methyl-3-pheny...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601050BDBM601050(4-((S)-3-((R)-3-cyclopropyl-3-phenylpropanamido)-2...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601219BDBM601219(US11634396, Compound 158 | 4-((S)-3-((S)-4,4-dimet...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601115BDBM601115(US11634396, Compound 74 | 4-[(2S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601118BDBM601118(US11634396, Compound 77 | 4-((S)-2-(dimethylamino)...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601224BDBM601224(US11634396, Compound 161 | 44-((S)-2-(1H-imidazol-...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601313BDBM601313((S)-3-cyclopropyl-N-((S)-2-(dimethylamino)-3-(4-hy...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601224BDBM601224(US11634396, Compound 161 | 44-((S)-2-(1H-imidazol-...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601117BDBM601117(US11634396, Compound 76 | 4-[(2S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601226BDBM601226(US11634396, Compound 163 | 4-((S)-2-(dimethylamino...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601119BDBM601119(US11634396, Compound 78 | 4-[(2S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetKappa-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601317BDBM601317((R)-N-((S)-2-(dimethylamino)-3-(4-hydroxy-2-(trifl...)
Affinity DataIC50: 300nMAssay Description:KOR β-Arrestin Agonist and Antagonist assays were preformed using the Tango OPRK1-bla U2OS cells from Invitrogen and purchased from ThermoFisher...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601227BDBM601227(US11634396, Compound 164 | 4-((S)-2-(dimethylamino...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601137BDBM601137(US11634396, Compound 98 | 4-((S)-2-(dimethylamino)...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetDelta-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601254BDBM601254((R)-N-((S)-3-(4-chloro-1H-indazol-5-yl)-2-(dimethy...)
Affinity DataEC50: <300nMAssay Description:The dOR cAMP agonist and antagonist assays were conducted in a manner similar as described above for the mOR assays using CHO Tag-lite human dOR stab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601062BDBM601062(3-chloro-4-((S)-3-((R)-3-(pyridin-3-yl)-3-(1-(trif...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Epiodyne

US Patent
LigandChemical structure of BindingDB Monomer ID 601141BDBM601141(US11634396, Compound 103 | (R)-N-((S)-2-(dimethyla...)
Affinity DataIC50: 300nMAssay Description:CHO Tag-lite human mOR stable cell line from Cisbio (NCBI accession number: NM_000914.3, Bedford, Mass.) were seeded and grown to approximately 80% c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2023
Entry Details
US Patent

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