Compile Data Set for Download or QSAR
Report error Found 228 Enz. Inhib. hit(s) with all data for entry = 11253
LigandChemical structure of BindingDB Monomer ID 602903BDBM602903(US11649237, Example 125 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602919BDBM602919(US11649237, Example 141 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602916BDBM602916(US11649237, Example 138 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602907BDBM602907(US11649237, Example 129 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602904BDBM602904(US11649237, Example 126 | 1-(4-(8-amino-3-ethyl-5-...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602927BDBM602927(US11649237, Example 149 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602926BDBM602926(US11649237, Example 148 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602908BDBM602908(US11649237, Example 130 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602924BDBM602924(US11649237, Example 146 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602929BDBM602929(US11649237, Example 151 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 1nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602932BDBM602932(US11649237, Example 154 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602843BDBM602843(US11649237, Example 65 | 2-(4-(8-amino-3-isopropyl...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602939BDBM602939(US11649237, Example 161 | 1-(4-((4,6-difluoro-1H-b...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602920BDBM602920(US11649237, Example 142 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602847BDBM602847(US11649237, Example 69 | 2-(4-(8-amino-3-isopropyl...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602845BDBM602845(US11649237, Example 67 | 2-(4-(8-amino-3-isopropyl...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602947BDBM602947(US11649237, Example 169 | N-(4-(8-Amino-3-isopropy...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602849BDBM602849(US11649237, Example 71 | 2-(4-(8-amino-3-isopropyl...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602848BDBM602848(US11649237, Example 70 | 2-(4-(8-amino-3-isopropyl...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602928BDBM602928(US11649237, Example 150 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 2nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602934BDBM602934(US11649237, Example 156 | 3-Isopropyl-1-(4-((7-met...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602918BDBM602918(US11649237, Example 140 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602884BDBM602884(US11649237, Example 106 | 3-(4-{8-amino-3-ethyl-5-...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602943BDBM602943(US11649237, Example 165 | 1-(4-((7-fluoro-1H-benzo...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602941BDBM602941(US11649237, Example 163 | 3-isopropyl-1-(4-((5-met...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 603005BDBM603005(US11649237, Example 227 | N-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602899BDBM602899(US11649237, Example 121 | 1-(4-(8-Amino-3-isopropy...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602914BDBM602914(US11649237, Example 136 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602930BDBM602930(US11649237, Example 152 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 3nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602923BDBM602923(US11649237, Example 145 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 4nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602842BDBM602842(US11649237, Example 64 | 2-(4-(8-amino-3-isopropyl...)
Affinity DataIC50: 4nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602906BDBM602906(US11649237, Example 128 | 1-(5-(8-amino-3-isopropy...)
Affinity DataIC50: 4nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602942BDBM602942(US11649237, Example 164 | 2-((4-(8-amino-3-isoprop...)
Affinity DataIC50: 4nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602974BDBM602974(US11649237, Example 195 | N-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 4nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 603006BDBM603006(US11649237, Example 230 | N-(4-(8-amino-5-(4-((2-f...)
Affinity DataIC50: 4nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602853BDBM602853(US11649237, Example 75 | 2-(4-(8-amino-3-isopropyl...)
Affinity DataIC50: 5nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602965BDBM602965(US11649237, Example 186 | N-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 5nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602922BDBM602922(US11649237, Example 144 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 5nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602921BDBM602921(US11649237, Example 143 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 5nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602940BDBM602940(US11649237, Example 162 | 1-(4-((4,6-dimethyl-1H-b...)
Affinity DataIC50: 5nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602964BDBM602964(US11649237, Example 185 | N-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 5nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602863BDBM602863(US11649237, Example 85 | 1-(4-(8-amino-5-(4-aminoc...)
Affinity DataIC50: 6nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602902BDBM602902(US11649237, Example 124 | 1-(5-(8-amino-3-isopropy...)
Affinity DataIC50: 7nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602997BDBM602997(US11649237, Example 218 | N-(4-{8-amino-5-[4-(meth...)
Affinity DataIC50: 7nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602925BDBM602925(US11649237, Example 147 | 1-(4-(8-amino-3-methyl-5...)
Affinity DataIC50: 7nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602860BDBM602860(US11649237, Example 82 | 2-(5-(8-amino-3-isopropyl...)
Affinity DataIC50: 7nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602913BDBM602913(US11649237, Example 135 | 1-(4-(8-amino-3-isopropy...)
Affinity DataIC50: 7nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602945BDBM602945(US11649237, Example 167 | 1-(4-((7-chloro-1H-benzo...)
Affinity DataIC50: 7nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602875BDBM602875(US11649237, Example 97 | 3-{4-[8-amino-5-(4-aminoc...)
Affinity DataIC50: 8nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 602859BDBM602859(US11649237, Example 81 | 2-(5-(8-amino-3-isopropyl...)
Affinity DataIC50: 8nMAssay Description:The kinase reactions were performed in 384 well white ProxiPlate-384 Plus plates (PERKIN Elmer 6008280) using 25 mM MOPS assay buffer with 1 mM dithi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
US Patent

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