Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 11335
TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608309BDBM608309(US11691981, Compound 66)
Affinity DataIC50: 4nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608284BDBM608284(US11691981, Compound 41)
Affinity DataIC50: 12nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608255BDBM608255(US11691981, Compound 17)
Affinity DataIC50: 12nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608288BDBM608288(US11691981, Compound 45)
Affinity DataIC50: 13nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608336BDBM608336(US11691981, Compound 73)
Affinity DataIC50: 14nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608308BDBM608308(US11691981, Compound 65)
Affinity DataIC50: 14nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 50564603BDBM50564603(CHEMBL4777294 | US11691981, Compound 77)
Affinity DataIC50: 17nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608337BDBM608337(US11691981, Compound 74)
Affinity DataIC50: 17nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608296BDBM608296(US11691981, Compound 53)
Affinity DataIC50: 18nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608281BDBM608281(US11691981, Compound 38)
Affinity DataIC50: 18nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608271BDBM608271(US11691981, Compound 29)
Affinity DataIC50: 19nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608295BDBM608295(US11691981, Compound 52)
Affinity DataIC50: 21nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608300BDBM608300(US11691981, Compound 57)
Affinity DataIC50: 21nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 50564620BDBM50564620(Ly-3200882 | Ly3200882 | US11691981, Compound A)
Affinity DataIC50: 22nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608341BDBM608341(US11691981, Compound 78)
Affinity DataIC50: 22nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608247BDBM608247(US11691981, Compound 11)
Affinity DataIC50: 24nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608314BDBM608314(US11691981, Compound 71)
Affinity DataIC50: 25nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608248BDBM608248(US11691981, Compound 12)
Affinity DataIC50: 28nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608342BDBM608342(US11691981, Compound 79)
Affinity DataIC50: 29nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608305BDBM608305(US11691981, Compound 62)
Affinity DataIC50: 29nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608302BDBM608302(US11691981, Compound 59)
Affinity DataIC50: 32nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608292BDBM608292(US11691981, Compound 49)
Affinity DataIC50: 32nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608307BDBM608307(US11691981, Compound 64)
Affinity DataIC50: 32nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608254BDBM608254(US11691981, Compound 16)
Affinity DataIC50: 34nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608298BDBM608298(US11691981, Compound 55)
Affinity DataIC50: 35nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608269BDBM608269(US11691981, Compound 28)
Affinity DataIC50: 35nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608261BDBM608261(US11691981, Compound 21)
Affinity DataIC50: 37nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608250BDBM608250(US11691981, Compound 14)
Affinity DataIC50: 37nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608263BDBM608263(US11691981, Compound 23)
Affinity DataIC50: 38nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608301BDBM608301(US11691981, Compound 58)
Affinity DataIC50: 39nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608277BDBM608277(US11691981, Compound 34)
Affinity DataIC50: 42nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608239BDBM608239(US11691981, Compound 5)
Affinity DataIC50: 43nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608249BDBM608249(US11691981, Compound 13)
Affinity DataIC50: 44nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608240BDBM608240(US11691981, Compound 6)
Affinity DataIC50: 46nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608260BDBM608260(US11691981, Compound 20)
Affinity DataIC50: 48nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608276BDBM608276(US11691981, Compound 33)
Affinity DataIC50: 49nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608303BDBM608303(US11691981, Compound 60)
Affinity DataIC50: 50nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608310BDBM608310(US11691981, Compound 67)
Affinity DataIC50: 51nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608343BDBM608343(US11691981, Compound 80 | US11691981, Compound 81)
Affinity DataIC50: 51nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608235BDBM608235(US11691981, Compound 2)
Affinity DataIC50: 53nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608262BDBM608262(US11691981, Compound 22)
Affinity DataIC50: 54nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608294BDBM608294(US11691981, Compound 51)
Affinity DataIC50: 55nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608279BDBM608279(US11691981, Compound 36)
Affinity DataIC50: 56nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608297BDBM608297(US11691981, Compound 54)
Affinity DataIC50: 56nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608343BDBM608343(US11691981, Compound 80 | US11691981, Compound 81)
Affinity DataIC50: 57nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608241BDBM608241(US11691981, Compound 7 | US11691981, Compound 27)
Affinity DataIC50: 58nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608238BDBM608238(US11691981, Compound 4)
Affinity DataIC50: 60nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608234BDBM608234(US11691981, Compound 1)
Affinity DataIC50: 61nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608265BDBM608265(US11691981, Compound 25)
Affinity DataIC50: 66nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandChemical structure of BindingDB Monomer ID 608289BDBM608289(US11691981, Compound 46)
Affinity DataIC50: 66nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
US Patent

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