Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 11559
TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 328995BDBM328995(US9663503, Compound Y-154 | 1137478-47-7 | US11787...)
Affinity DataIC50: 1nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 328993BDBM328993(US9663503, Compound 1 | 5-[[4-[[(2R)-morpholin-2-y...)
Affinity DataIC50: 1.40nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 328996BDBM328996(US9663503, Compound Y-081 | 1137477-07-6 | US11787...)
Affinity DataIC50: 2nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 328997BDBM328997(US9663503, Compound Y-152 | 1137478-45-5 | US11787...)
Affinity DataIC50: 2nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 328998BDBM328998(US9663503, Compound Y-158 | 1137478-52-4 | US11787...)
Affinity DataIC50: 2nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 328994BDBM328994(US9663503, Compound 2 | 5-[[4-[[(2S)-morpholin-2-y...)
Affinity DataIC50: 2.10nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 328999BDBM328999(US9663503, Compound Y-147 | 1137478-38-6 | US11787...)
Affinity DataIC50: 4nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329000BDBM329000(US9663503, Compound Y-153 | 1137478-46-6 | US11787...)
Affinity DataIC50: 4nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329001BDBM329001(US9663503, Compound Y-155 | 1137478-48-8 | US11787...)
Affinity DataIC50: 5nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329002BDBM329002(US9663503, Compound Y-149 | 1137478-40-0 | US11787...)
Affinity DataIC50: 10nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329003BDBM329003(US9663503, Compound Y-156 | 1137478-50-2 | US11787...)
Affinity DataIC50: 10nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329004BDBM329004(US9663503, Compound Y-146 | 1168103-91-0 | US11787...)
Affinity DataIC50: 11nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329005BDBM329005(US9663503, Compound Y-148 | 1137478-39-7 | US11787...)
Affinity DataIC50: 13nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329006BDBM329006(US9663503, Compound Y-157 | 1137478-51-3 | US11787...)
Affinity DataIC50: 15nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329007BDBM329007(US9663503, Compound Y-150 | 1137478-41-1 | US11787...)
Affinity DataIC50: 17nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329008BDBM329008(US9663503, Compound Y-102 | 1137477-35-0 | US11787...)
Affinity DataIC50: 20nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329009BDBM329009(US9663503, Compound Y-159 | 1137478-54-6 | US11787...)
Affinity DataIC50: 23nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk1(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 329010BDBM329010(US9663503, Compound Y-151 | 1137478-44-4 | US11787...)
Affinity DataIC50: 24nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent