Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 11692
TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640362BDBM640362(Preparation of 3-((8-amino-3-isopropylimidazo[1,5-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640363BDBM640363(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640363BDBM640363(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640364BDBM640364(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640361BDBM640361(Preparation of 3-((8-amino-3-methylimidazo[1,5-a]p...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640361BDBM640361(Preparation of 3-((8-amino-3-methylimidazo[1,5-a]p...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640362BDBM640362(Preparation of 3-((8-amino-3-isopropylimidazo[1,5-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640366BDBM640366(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640367BDBM640367(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640367BDBM640367(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640364BDBM640364(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640365BDBM640365(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640366BDBM640366(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640359BDBM640359(Preparation of 3-((8-amino-3-ethylimidazo[1,5-a]py...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640359BDBM640359(Preparation of 3-((8-amino-3-ethylimidazo[1,5-a]py...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640379BDBM640379(Preparation of N-(3-((4-amino-7-ethyl-7H-pyrrolo[2...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640380BDBM640380(Preparation of 3-((4-amino-7-((1r,4r)-4-hydroxycyc...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640376BDBM640376(Preparation of N-(3-((4-amino-7-ethyl-7H-pyrrolo[2...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640377BDBM640377(Preparation of N-(3-((4-amino-7-methyl-7H-pyrrolo[...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640377BDBM640377(Preparation of N-(3-((4-amino-7-methyl-7H-pyrrolo[...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640383BDBM640383(Preparation of N-(3-((4-amino-7-((1r,4r)-4-hydroxy...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640383BDBM640383(Preparation of N-(3-((4-amino-7-((1r,4r)-4-hydroxy...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640380BDBM640380(Preparation of 3-((4-amino-7-((1r,4r)-4-hydroxycyc...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640381BDBM640381(Preparation of 3-((4-amino-7-((1r,4r)-4-hydroxycyc...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640382BDBM640382(Preparation of 3-((4-amino-7-((1r,4r)-4-hydroxycyc...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640372BDBM640372(Preparation of 3-((4-amino-7-methyl-7H-pyrrolo[2,3...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640369BDBM640369(Preparation of 3-((4-amino-7-methyl-7H-pyrrolo[2,3...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640374BDBM640374(Preparation of 3-((4-amino-7-methyl-7H-pyrrolo[2,3...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640375BDBM640375(Preparation of N-(3-((4-amino-7-ethyl-7H-pyrrolo[2...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640375BDBM640375(Preparation of N-(3-((4-amino-7-ethyl-7H-pyrrolo[2...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640376BDBM640376(Preparation of N-(3-((4-amino-7-ethyl-7H-pyrrolo[2...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640372BDBM640372(Preparation of 3-((4-amino-7-methyl-7H-pyrrolo[2,3...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640373BDBM640373(Preparation of 3-((4-amino-7-isopropyl-7H-pyrrolo[...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640373BDBM640373(Preparation of 3-((4-amino-7-isopropyl-7H-pyrrolo[...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640374BDBM640374(Preparation of 3-((4-amino-7-methyl-7H-pyrrolo[2,3...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640379BDBM640379(Preparation of N-(3-((4-amino-7-ethyl-7H-pyrrolo[2...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640378BDBM640378(Preparation of N-(3-((4-amino-7-cyclopentyl-7H-pyr...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640382BDBM640382(Preparation of 3-((4-amino-7-((1r,4r)-4-hydroxycyc...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640368BDBM640368(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640365BDBM640365(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640381BDBM640381(Preparation of 3-((4-amino-7-((1r,4r)-4-hydroxycyc...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640370BDBM640370(Preparation of 3-((4-amino-7-isopropyl-7H-pyrrolo[...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640371BDBM640371(Preparation of 3-((4-amino-7-isopropyl-7H-pyrrolo[...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640371BDBM640371(Preparation of 3-((4-amino-7-isopropyl-7H-pyrrolo[...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640368BDBM640368(Preparation of 3-((4-amino-7-ethyl-7H-pyrrolo[2,3-...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640369BDBM640369(Preparation of 3-((4-amino-7-methyl-7H-pyrrolo[2,3...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640370BDBM640370(Preparation of 3-((4-amino-7-isopropyl-7H-pyrrolo[...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640360BDBM640360(Preparation of 3-((8-amino-3-ethylimidazo[1,5-a]py...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640378BDBM640378(Preparation of N-(3-((4-amino-7-cyclopentyl-7H-pyr...)
Affinity DataIC50: 75nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640360BDBM640360(Preparation of 3-((8-amino-3-ethylimidazo[1,5-a]py...)
Affinity DataIC50: 75nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent