Compile Data Set for Download or QSAR
Report error Found 328 Enz. Inhib. hit(s) with all data for entry = 11775
TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646150BDBM646150(US11878965, Example 206 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 13nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646149BDBM646149(US11878965, Example 134 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 18.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646246BDBM646246(US11878965, Example 237 | (R)-N-((R)-1-(2-(5-((1R,...)
Affinity DataIC50: 18.5nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646113BDBM646113(US11878965, Example 98 | ((1R,2R,4S)-2-amino-7- az...)
Affinity DataIC50: 18.9nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646118BDBM646118(US11878965, Example 103 | ((1R,2R,4S)-2-amino-7- a...)
Affinity DataIC50: 22.3nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646146BDBM646146(US11878965, Example 131 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 25.9nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646155BDBM646155(US11878965, Example 140 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 26.1nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646153BDBM646153(US11878965, Example 138 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 27.6nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646138BDBM646138(US11878965, Example 136 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 27.6nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646114BDBM646114(US11878965, Example 99 | ((R)-3-aminopiperidin-1-y...)
Affinity DataIC50: 28.4nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646247BDBM646247(US11878965, Example 238 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 28.7nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646195BDBM646195(US11878965, Example 180 | N-((R)-1-(2-(5-((R)-5-am...)
Affinity DataIC50: 28.8nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646154BDBM646154(US11878965, Example 139 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 28.9nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646138BDBM646138(US11878965, Example 136 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 29.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646120BDBM646120(US11878965, Example 105 | ((R)-3-aminopiperidin-1-...)
Affinity DataIC50: 29.6nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646254BDBM646254(US11878965, Example 245 | 1-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 31.7nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646136BDBM646136(N-((R)-1-(2-(5-((1R,2R,4S)-2- amino-7-azabicyclo[2...)
Affinity DataIC50: 32.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646094BDBM646094(US11878965, Example 79 | N-(2-(5-((1R,2R,4S)-2- am...)
Affinity DataIC50: 33.6nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646243BDBM646243(US11878965, Example 234 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 34.3nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646129BDBM646129(US11878965, Example 114 | methyl (2-(5-((1R,2R,4S)...)
Affinity DataIC50: 34.5nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646071BDBM646071(US11878965, Example 56 | N-(2-(5-((1R,2R,5R)-2-ami...)
Affinity DataIC50: 36.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646256BDBM646256(US11878965, Example 247 | 1-((R)-2-(2-(5-((1R,2R,4...)
Affinity DataIC50: 36.7nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646139BDBM646139(N-((R)-1-(2-(5-((R)-3- aminopiperidine-1-carbonyl)...)
Affinity DataIC50: 37.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646069BDBM646069(US11878965, Example 54 | (R)-N-(2-(5-(3-aminopiper...)
Affinity DataIC50: 37.4nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646264BDBM646264(US11878965, Example 255 | 1-(2-(5-((1R,2R,4S)-2-am...)
Affinity DataIC50: 40.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646244BDBM646244(US11878965, Example 235 | 3-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 40.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646257BDBM646257(US11878965, Example 248 | ((R)-2-(2-(5-((1R,2R,4S)...)
Affinity DataIC50: 40.5nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646117BDBM646117(US11878965, Example 102 | ((1R,2R,4S)-2-amino-7- a...)
Affinity DataIC50: 42nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646116BDBM646116(US11878965, Example 101 | ((R)-3-aminopiperidin-1-...)
Affinity DataIC50: 43.4nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646157BDBM646157(US11878965, Example 142 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 44.5nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646189BDBM646189(US11878965, Example 174 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 45.1nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646078BDBM646078(US11878965, Example 63 | N-(2-(5-((1R,2R,4S)-2- am...)
Affinity DataIC50: 45.1nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646145BDBM646145(US11878965, Example 130 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 45.1nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646150BDBM646150(US11878965, Example 206 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 45.5nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646133BDBM646133(US11878965, Example 118 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 45.6nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646161BDBM646161(US11878965, Example 146 | N-((R)-2-(2-(5-((1R,2R,4...)
Affinity DataIC50: 45.8nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646136BDBM646136(N-((R)-1-(2-(5-((1R,2R,4S)-2- amino-7-azabicyclo[2...)
Affinity DataIC50: 46.3nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646239BDBM646239(US11878965, Example 227 | (R)-N-((R)-1-(2-(5-((1S,...)
Affinity DataIC50: 46.8nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646080BDBM646080(US11878965, Example 65 | N-(2-(5-((1R,2R,4S)-2- am...)
Affinity DataIC50: 47nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646219BDBM646219(US11878965, Example 204 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 47.4nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646184BDBM646184(US11878965, Example 169 | N-((R)-1-(2-(5-((R)-5-am...)
Affinity DataIC50: 47.8nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646236BDBM646236(US11878965, Example 224 | N-((R)-1-(2-(5-((1S,4R,5...)
Affinity DataIC50: 48.1nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646237BDBM646237(US11878965, Example 225 | N-((R)-1-(2-(5-((1S,4R,5...)
Affinity DataIC50: 48.1nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646255BDBM646255(US11878965, Example 246 | 1-((R)-2-(2-(5-((1R,2R,4...)
Affinity DataIC50: 48.4nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646316BDBM646316(US11878965, Example 304 | N-((R)-1-(2-(5-((1S,4R,5...)
Affinity DataIC50: 48.6nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646253BDBM646253(US11878965, Example 244 | 1-((R)-1-(2-(5-((R)-3- a...)
Affinity DataIC50: 49.3nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646245BDBM646245(US11878965, Example 236 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 51.3nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646252BDBM646252(US11878965, Example 243 | N-((R)-1-(2-(5-((1R,2R,4...)
Affinity DataIC50: 52.8nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646238BDBM646238(US11878965, Example 226 | (S)-N-((R)-1-(2-(5-((1S,...)
Affinity DataIC50: 53.2nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

TargetProtein-arginine deiminase type-4(Human)
Gilead Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 646234BDBM646234(US11878965, Example 222 | N-((R)-1-(2-(5-((1S,4R,5...)
Affinity DataIC50: 53.5nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2024
Entry Details
US Patent

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