Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 11836
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651973BDBM651973(2-(4-((2′-methyl-[1,1′-biphenyl]-3-met...)
Affinity DataEC50:  4.80nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651977BDBM651977(2-(4-((2′-trifluoromethyl-[1,1′-biphen...)
Affinity DataEC50:  11.7nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651978BDBM651978(2-(4-((4′-ethoxy-2′-methyl-[1,1′...)
Affinity DataEC50:  14.6nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651970BDBM651970(2-(4-((2′-chloro-[1,1′-biphenyl]-3-met...)
Affinity DataEC50:  16.3nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651974BDBM651974(2-(4-((2′-methyl-[1,1′-biphenyl]-3-met...)
Affinity DataEC50:  17.3nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651976BDBM651976(2-(4-((2′-trifluoromethyl-[1,1′-biphen...)
Affinity DataEC50:  17.9nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651981BDBM651981(2-(4-(((4′-methoxy-2′-methyl-[1,1̸...)
Affinity DataEC50:  18.4nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651972BDBM651972(2-(4-((2′-chloro-[1,1′-biphenyl]-3-met...)
Affinity DataEC50:  18.6nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651969BDBM651969(2-(4-((4′-ethoxy-2′,6′-dimethyl-...)
Affinity DataEC50:  24.2nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 651980BDBM651980(2-(4-((4′-propoxy-2′-methyl-[1,1′...)
Affinity DataEC50:  28.4nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

US Patent
LigandChemical structure of BindingDB Monomer ID 50386790BDBM50386790(CHEMBL1829174 | CHEMBL2047159 | TAK-875 | US119052...)
Affinity DataEC50:  37.1nMAssay Description:hGPR40-CHO stably transfected cells were seeded into a 96-well plate at a density of 3×104/well, and incubated overnight in a 37° C., 5% CO2 cell inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
US Patent