Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 11867
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655581BDBM655581(US11912737, Example 31.)
Affinity DataIC50: 30nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655561BDBM655561(US11912737, Example 1 | US11912737, Example 7.)
Affinity DataIC50: 30nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655564BDBM655564(US11912737, Example 2 | US11912737, Example 10.)
Affinity DataIC50: 75nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655577BDBM655577(US11912737, Example 25.)
Affinity DataIC50: 75nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655603BDBM655603(US11912737, Example 53.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655602BDBM655602(US11912737, Example 52.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655570BDBM655570(US11912737, Example 18.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655573BDBM655573(US11912737, Example 21.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655572BDBM655572(US11912737, Example 20.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655567BDBM655567(US11912737, Example 13.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655575BDBM655575(US11912737, Example 51. | US11912737, Example 23.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655579BDBM655579(US11912737, Example 27.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655574BDBM655574(US11912737, Example 22.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655587BDBM655587(US11912737, Example 37.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655555BDBM655555(US11912737, Example 1.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655586BDBM655586(US11912737, Example 36.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655589BDBM655589(US11912737, Example 39.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655583BDBM655583(US11912737, Example 33.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655562BDBM655562(US11912737, Example 8.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655565BDBM655565(US11912737, Example 3 | US11912737, Example 11.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655558BDBM655558(US11912737, Example 4.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655560BDBM655560(US11912737, Example 6.)
Affinity DataIC50: 100nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655599BDBM655599(US11912737, Example 49.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655598BDBM655598(US11912737, Example 48.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655600BDBM655600(US11912737, Example 50.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655588BDBM655588(US11912737, Example 38.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655582BDBM655582(US11912737, Example 32.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655580BDBM655580(US11912737, Example 35. | US11912737, Example 28.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655584BDBM655584(US11912737, Example 34.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655595BDBM655595(US11912737, Example 45.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655594BDBM655594(US11912737, Example 44.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655597BDBM655597(US11912737, Example 47.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655596BDBM655596(US11912737, Example 46.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655591BDBM655591(US11912737, Example 41.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655590BDBM655590(US11912737, Example 40.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655593BDBM655593(US11912737, Example 43.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655592BDBM655592(US11912737, Example 42.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655571BDBM655571(US11912737, Example 19.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655566BDBM655566(US11912737, Example 12.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655569BDBM655569(US11912737, Example 17.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655568BDBM655568(US11912737, Example 15.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655578BDBM655578(US11912737, Example 26.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655580BDBM655580(US11912737, Example 35. | US11912737, Example 28.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655575BDBM655575(US11912737, Example 51. | US11912737, Example 23.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655576BDBM655576(US11912737, Example 24.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655557BDBM655557(US11912737, Example 3.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655556BDBM655556(US11912737, Example 2.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655563BDBM655563(US11912737, Example 9.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Sage Therpeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 655559BDBM655559(US11912737, Example 5.)
Affinity DataIC50: 500nMAssay Description:[35S]-t-Butylbicylophorothionate (TBPS) binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 655564BDBM655564(US11912737, Example 2 | US11912737, Example 10.)
Affinity DataEC50:  1.50E+3nMAssay Description:Whole cell currents were measured with HEKA EPC-10 amplifiers using PatchMaster software or by using the high throughput QPatch platform (Sophion). B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
US Patent

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