Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 12398
TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700723BDBM700723(US12115157, Ex. 13b)
Affinity DataEC50:  3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700715BDBM700715(US12115157, Ex. 8b)
Affinity DataEC50:  7nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700720BDBM700720(US12115157, Ex. 11b)
Affinity DataEC50:  10nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700728BDBM700728(BDBM700731 | (S)—N-(3-cyano-4-fluorophenyl)-1,2,4-...)
Affinity DataEC50:  11nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700725BDBM700725(US12115157, Ex. 14b)
Affinity DataEC50:  11nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700717BDBM700717(US12115157, Ex. 10a)
Affinity DataEC50:  14nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700707BDBM700707(US12115157, Ex. 1)
Affinity DataEC50:  15nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700710BDBM700710(US12115157, Ex. 4)
Affinity DataEC50:  18nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700716BDBM700716(US12115157, Ex. 9)
Affinity DataEC50:  19nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700726BDBM700726(US12115157, Ex. 15a)
Affinity DataEC50:  20nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700708BDBM700708(US12115157, Ex. 2)
Affinity DataEC50:  24nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700721BDBM700721(US12115157, Ex. 12)
Affinity DataEC50:  24nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700711BDBM700711(US12115157, Ex. 5)
Affinity DataEC50:  27nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700712BDBM700712(US12115157, Ex. 6)
Affinity DataEC50:  54nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700709BDBM700709(US12115157, Ex. 3)
Affinity DataEC50:  92nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700713BDBM700713(US12115157, Ex. 7)
Affinity DataEC50:  102nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700727BDBM700727(US12115157, Ex. 15b)
Affinity DataEC50:  168nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700729BDBM700729(US12115157, Ex. 16b)
Affinity DataEC50:  210nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700730BDBM700730(US12115157, Int. H-3)
Affinity DataEC50:  378nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700722BDBM700722(US12115157, Ex. 13a)
Affinity DataEC50:  595nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700714BDBM700714(US12115157, Ex. 8a)
Affinity DataEC50:  1.09E+3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700724BDBM700724(US12115157, Ex. 14a)
Affinity DataEC50:  1.17E+3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700719BDBM700719(US12115157, Ex. 11a)
Affinity DataEC50:  1.28E+3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent

TargetG-protein coupled receptor 52(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 700718BDBM700718(US12115157, Ex. 10b)
Affinity DataEC50:  1.33E+3nMAssay Description:HTRF cAMP assays were performed using commercially available assay kits according to the manufacturer's instructions (cAMP Dynamic 2 Assay Kit; #...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2025
Entry Details
US Patent