Compile Data Set for Download or QSAR
Report error Found 100 Enz. Inhib. hit(s) with all data for entry = 12411
TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701209BDBM701209(4-[2-(N-[(1S)-3,3-difluorocyclohexyl]anilino)- 2-o...)
Affinity DataKi:  0.114nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 50622931BDBM50622931(CHEMBL5409738 | US12122750, Example 44)
Affinity DataKi:  0.311nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 50622929BDBM50622929(CHEMBL5416925 | US12122750, Example 11)
Affinity DataKi:  0.336nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 50622932BDBM50622932(CHEMBL5400661 | US12122750, Example 53)
Affinity DataKi:  0.342nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 50622930BDBM50622930(CHEMBL5408779 | US12122750, Example 32)
Affinity DataKi:  0.345nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 50622927BDBM50622927(CHEMBL5430412 | US12122750, Example 2)
Affinity DataKi:  0.352nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 50622928BDBM50622928(CHEMBL5430333 | US12122750, Example 7)
Affinity DataKi:  0.382nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701241BDBM701241(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  0.383nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701184BDBM701184(4-[2-(N-cyclohexyl-3-fluoro-anilino)-2-oxo- ethyl]...)
Affinity DataKi:  0.400nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701213BDBM701213(4-[2-(2-fluoro-N-(2-fluorophenyl)anilino)-2- oxo-e...)
Affinity DataKi:  0.409nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701176BDBM701176(1-[methyl(phenyl)carbamoyl]-4-[2-oxo-2-(N- phenyla...)
Affinity DataKi:  0.428nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701218BDBM701218(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  0.471nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701169BDBM701169(4-[2-(N-cyclohexylanilino)-2-oxo-ethyl]-1-[(2- flu...)
Affinity DataKi:  0.521nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701179BDBM701179(1-[(4-fluorophenyl)-methyl-carbamoyl]-4-[2- (N-(3-...)
Affinity DataKi:  0.573nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701219BDBM701219(4-[2-(N-(3,3-difluorocyclohexyl)-2-fluoro- anilino...)
Affinity DataKi:  0.580nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701233BDBM701233(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  0.619nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701187BDBM701187(4-[2-(N-(4-fluorophenyl)anilino)-2-oxo-ethyl]- 1-[...)
Affinity DataKi:  0.716nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701181BDBM701181(4-[2-(N-(3-fluorophenyl)anilino)-2-oxo-ethyl]- 1-[...)
Affinity DataKi:  0.774nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701180BDBM701180(1-[(4-fluorophenyl)-methyl-carbamoyl]-4-[2- [N-(m-...)
Affinity DataKi:  0.823nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701208BDBM701208(4-[2-(N-[(1R)-3,3-difluorocyclohexyl]anilino)- 2-o...)
Affinity DataKi:  0.899nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701196BDBM701196(1-[(4-fluorophenyl)-methyl-carbamoyl]-4-[2- [N-(o-...)
Affinity DataKi:  0.987nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701194BDBM701194(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  1.03nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701231BDBM701231(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  1.04nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701229BDBM701229(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  1.04nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701239BDBM701239(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  1.09nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701230BDBM701230(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  1.19nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701243BDBM701243(4-(2-((3,3-difluorocyclohexyl)(phenyl)amino)- 2-ox...)
Affinity DataKi:  1.28nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701214BDBM701214(1-(6-cyanoindoline-1-carbonyl)-4-[2-(N-(3,3- diflu...)
Affinity DataKi:  1.34nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701199BDBM701199(1-[cyclopropyl-(4-fluorophenyl)carbamoyl]-4- [2-(N...)
Affinity DataKi:  1.37nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701217BDBM701217(1-[(4-cyclopropylphenyl)methyl]-4-[2-(N-(3,3- difl...)
Affinity DataKi:  1.38nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701170BDBM701170(4-[2-(N-cyclohexylanilino)-2-oxo-ethyl]-1- [methyl...)
Affinity DataKi:  1.44nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701211BDBM701211(1-[(4-cyclopropylphenyl)-methyl-carbamoyl]-4- [2-o...)
Affinity DataKi:  1.55nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701167BDBM701167(4-[2-(N-(2,2-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  1.56nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701172BDBM701172(4-[2-(N-cyclohexylanilino)-2-oxo-ethyl]-1- [ethyl-...)
Affinity DataKi:  1.69nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701173BDBM701173(4-[2-(N-cyclohexylanilino)-2-oxo-ethyl]-1- [cyclop...)
Affinity DataKi:  1.76nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701188BDBM701188(4-[2-(N-(4-chlorophenyl)anilino)-2-oxo-ethyl]- 1-[...)
Affinity DataKi:  1.89nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701190BDBM701190(1-(6-cyanoindoline-1-carbonyl)-4-[2-(N- cyclohexyl...)
Affinity DataKi:  1.94nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701221BDBM701221(4-[2-(N-(3,3-difluorocyclohexyl)-4-fluoro- anilino...)
Affinity DataKi:  2nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701177BDBM701177(4-[2-(N-(1-cyclopropylcyclopropyl)anilino)-2- oxo-...)
Affinity DataKi:  2.11nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701205BDBM701205(4-[2-[N-(1-cyclopropylethyl)anilino]-2-oxo- ethyl]...)
Affinity DataKi:  2.19nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701234BDBM701234(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  2.31nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701232BDBM701232(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  2.55nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701171BDBM701171(4-[2-(N-cyclohexylanilino)-2-oxo-ethyl]-1-[(4- met...)
Affinity DataKi:  2.58nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701166BDBM701166(4-[2-(N-cyclopentylanilino)-2-oxo-ethyl]-1-[(4- fl...)
Affinity DataKi:  2.62nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701212BDBM701212(1-[(4-cyclopropylphenyl)-methyl-carbamoyl]-4- [2-o...)
Affinity DataKi:  2.68nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701182BDBM701182(1-[(4-fluorophenyl)-methyl-carbamoyl]-4-[2- (N-(3-...)
Affinity DataKi:  2.70nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701192BDBM701192(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  2.79nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701198BDBM701198(1-[cyclopropyl-(4-fluorophenyl)carbamoyl]-4- [2-ox...)
Affinity DataKi:  2.82nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701235BDBM701235(4-[2-(N-(3,3-difluorocyclohexyl)anilino)-2- oxo-et...)
Affinity DataKi:  2.93nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 701204BDBM701204(4-[2-[N-(1-cyclopropylethyl)anilino]-2-oxo- ethyl]...)
Affinity DataKi:  2.93nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/24/2025
Entry Details
US Patent

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