Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 12751
LigandPNGBDBM725110(US12240839, Example 5)
Affinity DataIC50: 2nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725116(Cis-(P)-1-(5-Chloro-4-(3-Fluoro-3-(Trifluoromethyl...)
Affinity DataIC50: 2nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725114(Trans-(P)-1-(5-Fluoro-4-(3-Fluoro-3-(Trifluorometh...)
Affinity DataIC50: 2nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725146(US12240839, Example 40)
Affinity DataIC50: 5nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725113(Trans-(P)-1-(5-Fluoro-4-(3-Fluoro-3-(Trifluorometh...)
Affinity DataIC50: 5nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725118(US12240839, Example 13)
Affinity DataIC50: 6nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725148(US12240839, Example 42)
Affinity DataIC50: 6nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725117(Cis-(P)-1-(5-Chloro-2-Methoxy-4-(3-(Trifluoromethy...)
Affinity DataIC50: 7nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725149(US12240839, Example 43)
Affinity DataIC50: 7nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725150(1-(5-Fluoro-2-Methoxy-4-((1R,3R)-3-(Trifluorometho...)
Affinity DataIC50: 7nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725112(US12240839, Example 7)
Affinity DataIC50: 7nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725154(US12240839, Example 47)
Affinity DataIC50: 8nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725151(US12240839, Example 45)
Affinity DataIC50: 8nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725153(US12240839, Example 46)
Affinity DataIC50: 8nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725115(Cis-(P)-1-(5-Chloro-4-(3-Fluoro-3-(Trifluoromethyl...)
Affinity DataIC50: 8nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725136(US12240839, Example 32)
Affinity DataIC50: 10nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725156(US12240839, Example 49)
Affinity DataIC50: 10nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725155(US12240839, Example 48)
Affinity DataIC50: 10nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725145(US12240839, Example 39)
Affinity DataIC50: 11nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725111(Cis-(P)-1-(5-Fluoro-2-Methoxy-4-(3-(Trifluoromethy...)
Affinity DataIC50: 11nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725147(US12240839, Example 41)
Affinity DataIC50: 11nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725126(US12240839, Example 21)
Affinity DataIC50: 12nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725125(US12240839, Example 20)
Affinity DataIC50: 12nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725129(US12240839, Example 24)
Affinity DataIC50: 13nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725142(US12240839, Example 36)
Affinity DataIC50: 14nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725124(US12240839, Example 19)
Affinity DataIC50: 15nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725109(US12240839, Example 4)
Affinity DataIC50: 15nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725122(US12240839, Example 17)
Affinity DataIC50: 15nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725119(US12240839, Example 14)
Affinity DataIC50: 16nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725120(US12240839, Example 15)
Affinity DataIC50: 17nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725121(Cis-(P)-1-(5-Chloro-2-Methoxy-4-(3-(Trifluoromethy...)
Affinity DataIC50: 18nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725141(US12240839, Example 35)
Affinity DataIC50: 20nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725144(US12240839, Example 38)
Affinity DataIC50: 21nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725123(US12240839, Example 18)
Affinity DataIC50: 22nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725107(US12240839, Example 2)
Affinity DataIC50: 25nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725137(US12240839, Example 34)
Affinity DataIC50: 28nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725108(US12240839, Example 3)
Affinity DataIC50: 33nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725134(US12240839, Example 29)
Affinity DataIC50: 37nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725130(US12240839, Example 25)
Affinity DataIC50: 37nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM218114(US9212182, 1145 | US12240839, Compound X)
Affinity DataIC50: 48nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725127(US12240839, Example 22)
Affinity DataIC50: 50nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725133(US12240839, Example 28)
Affinity DataIC50: 54nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725143(US12240839, Example 37)
Affinity DataIC50: 62nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725131(US12240839, Example 26)
Affinity DataIC50: 80nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725128(US12240839, Example 23)
Affinity DataIC50: 102nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725132(US12240839, Example 27)
Affinity DataIC50: 104nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent

LigandPNGBDBM725135(US12240839, Example 30)
Affinity DataIC50: 137nMAssay Description:Human Nav1.7 currents were recorded in population patch-clamp mode with the IWB automated electrophysiology system (Molecular Devices, LLC, Sunnyvale...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
US Patent