Compile Data Set for Download or QSAR
Report error Found 237 Enz. Inhib. hit(s) with all data for entry = 13031
LigandPNGBDBM753477((S)-quinuclidin-3-yl (7-methoxy-2,2-dimethyl-6-(4-...)
Affinity DataIC50: 0.190nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753474((S)-quinuclidin-3-yl (7-fluoro-6-(4-isopropoxyphen...)
Affinity DataIC50: 0.290nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753472((S)-quinuclidin-3-yl (7-fluoro-6-(4-isobutylphenyl...)
Affinity DataIC50: 0.300nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753471((S)-quinuclidin-3-yl (7-fluoro-2,2-dimethyl-6-(4-p...)
Affinity DataIC50: 0.310nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753469((S)-quinuclidin-3-yl (7-fluoro-6-(3-fluoro-4-metho...)
Affinity DataIC50: 0.5nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753478((S)-quinuclidin-3-yl (6-(4-isobutylphenyl)-7-metho...)
Affinity DataIC50: 0.530nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753480((S)-quinuclidin-3-yl (6-(4-isopropoxyphenyl)-7-met...)
Affinity DataIC50: 0.550nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753462((S)-quinuclidin-3-yl (6'-(4-propoxyphenyl)-3',4'-d...)
Affinity DataIC50: 0.630nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753352((S)-quinuclidin-3-yl (6-(4-(2-methoxyethoxy)phenyl...)
Affinity DataIC50: 0.640nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753475((S)-quinuclidin-3-yl (6-(3-fluoro-4-methoxyphenyl)...)
Affinity DataIC50: 0.650nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753249((S)-quinuclidin-3-yl (6-(3-chlorophenyl)-1,2,3,4-t...)
Affinity DataIC50: 0.697nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753464((S)-quinuclidin-3-yl (6'-(4-propylphenyl)-3',4'-di...)
Affinity DataIC50: 0.75nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753333((S)-quinuclidin-3-yl (6-(3-chlorophenyl)-2,2-dimet...)
Affinity DataIC50: 0.810nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753368((S)-quinuclidin-3-yl (6-(3-fluoro-4-methoxyphenyl)...)
Affinity DataIC50: 0.830nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753337((S)-quinuclidin-3-yl (6-(2-chlorophenyl)-2,2-dimet...)
Affinity DataIC50: 0.850nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753473((S)-quinuclidin-3-yl (6-(2-(tert-butoxy)pyridin-4-...)
Affinity DataIC50: 0.860nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753339((S)-quinuclidin-3-yl (2,2-dimethyl-6-(2-(trifluoro...)
Affinity DataIC50: 0.860nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753387((S)-quinuclidin-3-yl (6-(3-fluoro-4-propoxyphenyl)...)
Affinity DataIC50: 0.870nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753468((S)-quinuclidin-3-yl (6'-(4-cyclopropylphenyl)-3',...)
Affinity DataIC50: 0.930nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM753355((S)-quinuclidin-3-yl (6-(4-(methoxymethoxy)phenyl)...)
Affinity DataIC50: 0.940nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753345((S)-quinuclidin-3-yl (6-(2,5-difluorophenyl)-2,2-d...)
Affinity DataIC50: 0.950nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753336((S)-quinuclidin-3-yl (6-(2-fluorophenyl)-2,2-dimet...)
Affinity DataIC50: 0.970nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753365((S)-quinuclidin-3-yl (6-(2-chloro-4-methoxyphenyl)...)
Affinity DataIC50: 0.970nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753248((S)-quinuclidin-3-yl (6-(3-fluorophenyl)-1,2,3,4-t...)
Affinity DataIC50: 0.989nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM753344((S)-quinuclidin-3-yl (6-(2,3-difluorophenyl)-2,2-d...)
Affinity DataIC50: 1nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753389((S)-quinuclidin-3-yl (6-(4-butoxy-3,5-dimethylphen...)
Affinity DataIC50: 1nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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In Depth
Date in BDB:
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US Patent

LigandPNGBDBM753332((S)-quinuclidin-3-yl (6-(3-fluorophenyl)-2,2-dimet...)
Affinity DataIC50: 1.01nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM753459((S)-quinuclidin-3-yl (6'-(4-ethoxyphenyl)-3',4'-di...)
Affinity DataIC50: 1.01nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM753436((S)-quinuclidin-3-yl (6'-(4-(2-methoxyethoxy)pheny...)
Affinity DataIC50: 1.03nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
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US Patent

LigandPNGBDBM753334((S)-quinuclidin-3-yl (2,2-dimethyl-6-(3-(trifluoro...)
Affinity DataIC50: 1.04nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM753375((S)-quinuclidin-3-yl (6-(2,3-dimethoxyphenyl)-2,2-...)
Affinity DataIC50: 1.05nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM753367((S)-quinuclidin-3-yl (6-(2-chloro-5-methoxyphenyl)...)
Affinity DataIC50: 1.10nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753461((S)-quinuclidin-3-yl (6'-(4-isopropoxyphenyl)-3',4...)
Affinity DataIC50: 1.10nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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In Depth
Date in BDB:
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US Patent

LigandPNGBDBM753384((S)-quinuclidin-3-yl (6-(3-fluoro-4-isopropoxyphen...)
Affinity DataIC50: 1.11nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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In Depth
Date in BDB:
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US Patent

LigandPNGBDBM753444((S)-quinuclidin-3-yl (6'-(3-fluoro-4-methoxyphenyl...)
Affinity DataIC50: 1.16nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM753374((S)-quinuclidin-3-yl (6-(3-isopropoxyphenyl)-2,2-d...)
Affinity DataIC50: 1.16nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM753357((S)-quinuclidin-3-yl (6-(2-(methoxymethoxy)phenyl)...)
Affinity DataIC50: 1.17nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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In Depth
Date in BDB:
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LigandPNGBDBM753380((S)-quinuclidin-3-yl (6-(3,5-dimethoxyphenyl)-2,2-...)
Affinity DataIC50: 1.19nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM753372((S)-quinuclidin-3-yl (6-(3-(difluoromethyl)phenyl)...)
Affinity DataIC50: 1.24nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM753271((S)-quinuclidin-3-yl (6-(3-(methoxymethoxy)phenyl)...)
Affinity DataIC50: 1.33nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
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US Patent

LigandPNGBDBM753470((S)-quinuclidin-3-yl (6-(3,5-dimethyl-4-propoxyphe...)
Affinity DataIC50: 1.34nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753347((S)-quinuclidin-3-yl (6-(2,5-dichlorophenyl)-2,2-d...)
Affinity DataIC50: 1.39nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753386((S)-quinuclidin-3-yl (6-(4-ethoxy-3-fluorophenyl)-...)
Affinity DataIC50: 1.39nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753247((S)-quinuclidin-3-yl (6-(4-(trifluoromethoxy)pheny...)
Affinity DataIC50: 1.42nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753385((S)-quinuclidin-3-yl (6-(4-butoxy-3-chlorophenyl)-...)
Affinity DataIC50: 1.44nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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In Depth
Date in BDB:
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LigandPNGBDBM753476((S)-quinuclidin-3-yl (6-(3,5-dimethyl-4-propoxyphe...)
Affinity DataIC50: 1.45nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753382((S)-quinuclidin-3-yl (6-(3-chloro-4-ethoxyphenyl)-...)
Affinity DataIC50: 1.49nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753373((S)-quinuclidin-3-yl (6-(3-(dimethylamino)phenyl)-...)
Affinity DataIC50: 1.49nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753383((S)-quinuclidin-3-yl (6-(3-chloro-4-propoxyphenyl)...)
Affinity DataIC50: 1.51nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM753466((S)-quinuclidin-3-yl (6'-(4-isobutylphenyl)-3',4'-...)
Affinity DataIC50: 1.53nMAssay Description:(1) MaterialsA549 cells (ATCC, CCL-185)NBD C6-ceramide (Thermo Fisher, N1154)UDP-glucose (Sigma, U4625)Potassium chloride (Sigma, P9333)UltraPure™ 0....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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