Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 13033
TargetCytochrome P450 3A4(Human)
Teligene US

US Patent
LigandPNGBDBM50018830(CHEMBL3286830 | US10543199, Compound PF-06463922 |...)
Affinity DataIC50: 7.80E+3nMAssay Description:Human liver microsomes (HLM) are stored at −80° C. Before the study, microsomes were thawed in a cold water bath, and then were put on ice immediatel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2025
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Teligene US

US Patent
LigandPNGBDBM753489(US12338251, Compound 2)
Affinity DataIC50: 1.00E+4nMAssay Description:Human liver microsomes (HLM) are stored at −80° C. Before the study, microsomes were thawed in a cold water bath, and then were put on ice immediatel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/17/2025
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Teligene US

US Patent
LigandPNGBDBM753492(US12338251, Compound 3)
Affinity DataIC50: 2.79E+5nMAssay Description:Human liver microsomes (HLM) are stored at −80° C. Before the study, microsomes were thawed in a cold water bath, and then were put on ice immediatel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/17/2025
Entry Details
US Patent