Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 13118
LigandPNGBDBM760334(1-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- ...)
Affinity DataKi:  0.800nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760344(1-(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  1.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760333(1-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- ...)
Affinity DataKi:  1.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605888(CHEMBL5179759 | US12370182, Example 6)
Affinity DataKi:  2.70nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605882(CHEMBL5202280 | US12370182, Example 1)
Affinity DataKi:  2.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605904(CHEMBL5179688 | US12370182, Example 45)
Affinity DataKi:  3.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605868(CHEMBL5186978 | US12370182, Example 8)
Affinity DataKi:  3.70nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605891(CHEMBL5174560 | US12370182, Example 83)
Affinity DataKi:  3.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760297(4-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- ...)
Affinity DataKi:  4.30nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760345(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxolane-2-car...)
Affinity DataKi:  4.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605890(CHEMBL5200451 | US12370182, Example 3)
Affinity DataKi:  5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605894(CHEMBL5176630 | US12370182, Example 82)
Affinity DataKi:  5.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760338(2-fluoro-1-(2-{[1-(4- fluorophenyl)-4-methyl-1H- 1...)
Affinity DataKi:  5.30nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760346(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxolane-3-car...)
Affinity DataKi:  5.70nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605887(CHEMBL5193778 | US12370182, Example 9)
Affinity DataKi:  6.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760370(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- yl]...)
Affinity DataKi:  6.5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605886(CHEMBL5197478 | US12370182, Example 7)
Affinity DataKi:  6.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605885(CHEMBL5181374 | US12370182, Example 2)
Affinity DataKi:  7nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760331(cyclopropyl(2-{[1-(4- fluorophenyl)-4-methyl-1H- 1...)
Affinity DataKi:  7.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760352(1-(2-{[4-(4-chlorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  7.5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605883(CHEMBL5189320 | US12370182, Example 5)
Affinity DataKi:  7.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605892(CHEMBL5178153 | US12370182, Example 84)
Affinity DataKi:  8.90nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760354(2-fluoro-1-(2-{[4-(4- fluorophenyl)-1-methyl-1H- 1...)
Affinity DataKi:  9.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760347(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxane-3-carbo...)
Affinity DataKi:  9.5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760320(1-(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  9.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760295(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- yl]...)
Affinity DataKi:  11nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760337(2,2-difluoro-1-(2-{[1-(4- fluorophenyl)-4-methyl-1...)
Affinity DataKi:  11nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760339(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxane-4-carbo...)
Affinity DataKi:  13nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760326(1-(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  13nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760342(1-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  13nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760296(2,2,2-trifluoro-1-(2-{[3-(4- fluorophenyl)-5-methy...)
Affinity DataKi:  14nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760317(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  14nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760341(5-[({6-cyclobutanecarbonyl- 5H,6H,7H-pyrrolo[3,4- ...)
Affinity DataKi:  14nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605884(CHEMBL5193523 | US12370182, Example 4)
Affinity DataKi:  16nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760340(1-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  17nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760313(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  18nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760357(4-(4-fluorophenyl)-1-methyl- 5-({[6-(oxolane-2-car...)
Affinity DataKi:  18nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760322(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  18nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760351(1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760294(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- yl]...)
Affinity DataKi:  21nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760316(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  22nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760323(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  24nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760304(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  24nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760348(4-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  25nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760353(1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  25nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605901(CHEMBL5207798 | US12370182, Example 14)
Affinity DataKi:  28nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760349(3-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  28nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50605898(CHEMBL5184265 | US12370182, Example 78)
Affinity DataKi:  28nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760309(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  29nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760356(1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  29nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

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