Compile Data Set for Download or QSAR
Report error Found 1903 Enz. Inhib. hit(s) with all data for entry = 13119
LigandPNGBDBM760709(N-[3-fluoro-4-[[6-(2-methoxyethoxy)- 7-methyl-1,5-...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM760709(N-[3-fluoro-4-[[6-(2-methoxyethoxy)- 7-methyl-1,5-...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM760708(1-cyclopropyl-N-[3-fluoro-4-[(6- methoxy-1,5-napht...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM760708(1-cyclopropyl-N-[3-fluoro-4-[(6- methoxy-1,5-napht...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM760708(1-cyclopropyl-N-[3-fluoro-4-[(6- methoxy-1,5-napht...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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LigandPNGBDBM760707(1-cyclopropyl-N-[4-[(6,7-dimethoxy- 1,5-naphthyrid...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM760711(N-[3-fluoro-4-[[7-methyl-6-(3- morpholin-4-ylpropo...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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LigandPNGBDBM760711(N-[3-fluoro-4-[[7-methyl-6-(3- morpholin-4-ylpropo...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM760710(5-(4-fluorophenyl)-4-hydroxy-N-[4- [[6-(2-methoxye...)
Affinity DataIC50: 100nMAssay Description:Example B-1: Human KDR (residues K790-V1356, 55 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 0.33 mg/mL myelin basic protein, 10 mM magnesiu...More data for this Ligand-Target Pair
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LigandPNGBDBM760710(5-(4-fluorophenyl)-4-hydroxy-N-[4- [[6-(2-methoxye...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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LigandPNGBDBM760710(5-(4-fluorophenyl)-4-hydroxy-N-[4- [[6-(2-methoxye...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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LigandPNGBDBM760710(5-(4-fluorophenyl)-4-hydroxy-N-[4- [[6-(2-methoxye...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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LigandPNGBDBM760709(N-[3-fluoro-4-[[6-(2-methoxyethoxy)- 7-methyl-1,5-...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM760713(1-cyclopropyl-N-[4-[(6,7-dimethoxy- 1,5-naphthyrid...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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LigandPNGBDBM760713(1-cyclopropyl-N-[4-[(6,7-dimethoxy- 1,5-naphthyrid...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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LigandPNGBDBM760384(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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LigandPNGBDBM760712(1-cyclopropyl-N-[4-[(6,7-dimethoxy- 1,5-naphthyrid...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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LigandPNGBDBM760712(1-cyclopropyl-N-[4-[(6,7-dimethoxy- 1,5-naphthyrid...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM760711(N-[3-fluoro-4-[[7-methyl-6-(3- morpholin-4-ylpropo...)
Affinity DataIC50: 100nMAssay Description:Example B-1: Human KDR (residues K790-V1356, 55 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 0.33 mg/mL myelin basic protein, 10 mM magnesiu...More data for this Ligand-Target Pair
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Date in BDB:
TBA
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LigandPNGBDBM760711(N-[3-fluoro-4-[[7-methyl-6-(3- morpholin-4-ylpropo...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM760715(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM760715(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM760384(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760714(1-cyclopropyl-N-[3-fluoro-4-[(6- methoxy-1,5-napht...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760384(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760714(1-cyclopropyl-N-[3-fluoro-4-[(6- methoxy-1,5-napht...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760713(1-cyclopropyl-N-[4-[(6,7-dimethoxy- 1,5-naphthyrid...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
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US Patent

LigandPNGBDBM760717(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
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US Patent

LigandPNGBDBM760716(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example B-1: Human KDR (residues K790-V1356, 55 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 0.33 mg/mL myelin basic protein, 10 mM magnesiu...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760716(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
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US Patent

LigandPNGBDBM760716(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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Date in BDB:
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US Patent

LigandPNGBDBM760716(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760715(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example B-1: Human KDR (residues K790-V1356, 55 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 0.33 mg/mL myelin basic protein, 10 mM magnesiu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760715(N-[4-[(6,7-dimethoxy-1,5- naphthyridin-4-yl)oxy]-3...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760719(N-[3-fluoro-4-[(6-methoxy-7-prop-1- en-2-yl-1,5-na...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
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US Patent

LigandPNGBDBM760719(N-[3-fluoro-4-[(6-methoxy-7-prop-1- en-2-yl-1,5-na...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760718(5-(4-fluoro-2-methylphenyl)-4- hydroxy-6-methyl-N-...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760718(5-(4-fluoro-2-methylphenyl)-4- hydroxy-6-methyl-N-...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760718(5-(4-fluoro-2-methylphenyl)-4- hydroxy-6-methyl-N-...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760721(5-(4-fluorophenyl)-N-[3-fluoro-4-[(7- prop-1-en-2-...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760721(5-(4-fluorophenyl)-N-[3-fluoro-4-[(7- prop-1-en-2-...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM760720(5-(4-fluoro-2-methylphenyl)-N-[3- fluoro-4-[(7-pro...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
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Date in BDB:
TBA
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US Patent

LigandPNGBDBM760720(5-(4-fluoro-2-methylphenyl)-N-[3- fluoro-4-[(7-pro...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
TBA
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US Patent

LigandPNGBDBM760720(5-(4-fluoro-2-methylphenyl)-N-[3- fluoro-4-[(7-pro...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM760723(N-[3-fluoro-4-[(6-methoxy-7-prop-1- en-2-yl-1,5-na...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM760723(N-[3-fluoro-4-[(6-methoxy-7-prop-1- en-2-yl-1,5-na...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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Date in BDB:
TBA
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LigandPNGBDBM760722(N-[3-fluoro-4-[(6-methoxy-7-prop-1- en-2-yl-1,5-na...)
Affinity DataIC50: 100nMAssay Description:Example C-1: Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIY...More data for this Ligand-Target Pair
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Date in BDB:
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LigandPNGBDBM760722(N-[3-fluoro-4-[(6-methoxy-7-prop-1- en-2-yl-1,5-na...)
Affinity DataIC50: 100nMAssay Description:Example A-1: Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKSRGDYMTMQIG (SEQ ID NO:1), 1...More data for this Ligand-Target Pair
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Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760721(5-(4-fluorophenyl)-N-[3-fluoro-4-[(7- prop-1-en-2-...)
Affinity DataIC50: 100nMAssay Description:Example B-1: Human KDR (residues K790-V1356, 55 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 0.33 mg/mL myelin basic protein, 10 mM magnesiu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM760721(5-(4-fluorophenyl)-N-[3-fluoro-4-[(7- prop-1-en-2-...)
Affinity DataIC50: 100nMAssay Description:Example D-1: Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 M KKKGQEEEYVFIE (SE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TBA
Entry Details
US Patent

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