Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 13135
TargetCytochrome P450 1A2(Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM700731(US12115157, Ex. 16a | US12378192, Compound of form...)
Affinity DataIC50: 4.64E+4nMAssay Description:A final incubation system of 500 μL contained 50 μL of liver microsomes (protein concentration: 0.2 mg/mL, Corning), 1 μL of mixed specific substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent

TargetCytochrome P450 2C19(Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM700731(US12115157, Ex. 16a | US12378192, Compound of form...)
Affinity DataIC50: 6.00E+4nMAssay Description:A final incubation system of 500 μL contained 50 μL of liver microsomes (protein concentration: 0.2 mg/mL, Corning), 1 μL of mixed specific substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent

TargetCytochrome P450 2C9(Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM700731(US12115157, Ex. 16a | US12378192, Compound of form...)
Affinity DataIC50: 7.97E+4nMAssay Description:A final incubation system of 500 μL contained 50 μL of liver microsomes (protein concentration: 0.2 mg/mL, Corning), 1 μL of mixed specific substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent

TargetCytochrome P450 2B6(Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM700731(US12115157, Ex. 16a | US12378192, Compound of form...)
Affinity DataIC50: 1.46E+5nMAssay Description:A final incubation system of 500 μL contained 50 μL of liver microsomes (protein concentration: 0.2 mg/mL, Corning), 1 μL of mixed specific substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent

TargetCytochrome P450 3A4(Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM700731(US12115157, Ex. 16a | US12378192, Compound of form...)
Affinity DataIC50: 2.00E+5nMAssay Description:A final incubation system of 500 μL contained 50 μL of liver microsomes (protein concentration: 0.2 mg/mL, Corning), 1 μL of mixed specific substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent

TargetCytochrome P450 2D6(Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM700731(US12115157, Ex. 16a | US12378192, Compound of form...)
Affinity DataIC50: 2.24E+5nMAssay Description:A final incubation system of 500 μL contained 50 μL of liver microsomes (protein concentration: 0.2 mg/mL, Corning), 1 μL of mixed specific substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent