Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 13179
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765063(US12391669, Compound 47)
Affinity DataIC50: 10nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765075(US12391669, Compound 25)
Affinity DataIC50: 32nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765078(US12391669, Compound 20)
Affinity DataIC50: 52nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765079(US12391669, Compound 67)
Affinity DataIC50: 63nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765062(US12391669, Compound 96)
Affinity DataIC50: 98nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765075(US12391669, Compound 25)
Affinity DataIC50: 117nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765085(salt | US12391669, Compound 11)
Affinity DataIC50: 119nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765062(US12391669, Compound 96)
Affinity DataIC50: 120nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765063(US12391669, Compound 47)
Affinity DataIC50: 181nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765077(US12391669, Compound 16)
Affinity DataIC50: 228nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765074(US12391669, Compound 84)
Affinity DataIC50: 296nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765071(US12391669, Compound 30)
Affinity DataIC50: 439nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765081(US12391669, Compound 35)
Affinity DataIC50: 443nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765083(US12391669, Compound 51)
Affinity DataIC50: 524nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765076(US12391669, Compound 73)
Affinity DataIC50: 961nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765082(US12391669, Compound 39)
Affinity DataIC50: 1.14E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765076(US12391669, Compound 73)
Affinity DataIC50: 1.57E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765080(US12391669, Compound 43)
Affinity DataIC50: 1.60E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765074(US12391669, Compound 84)
Affinity DataIC50: 1.98E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765064(US12391669, Compound 77)
Affinity DataIC50: 2.10E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765084(US12391669, Compound 55)
Affinity DataIC50: 3.19E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765064(US12391669, Compound 77)
Affinity DataIC50: 6.20E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
University Of California

US Patent
LigandPNGBDBM765067(US12391669, Compound 88)
Affinity DataIC50: 7.30E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765071(US12391669, Compound 30)
Affinity DataIC50: 8.40E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765077(US12391669, Compound 16)
Affinity DataIC50: 1.00E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765078(US12391669, Compound 20)
Affinity DataIC50: 1.00E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE2(Human)
University Of California

US Patent
LigandPNGBDBM765067(US12391669, Compound 88)
Affinity DataIC50: 1.00E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent