Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 13369
TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783875(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.120nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783872(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.200nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783872(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.260nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783858(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.260nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783879(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.340nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783878(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.360nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783873(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.370nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783873(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.430nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783870(N-(Cis-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-1-...)
Affinity DataIC50: 0.430nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783871(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.430nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783877(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.470nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783867(1-(Cis-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-1-...)
Affinity DataIC50: 0.570nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783876(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.600nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783875(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.630nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783881(N-(4-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)e...)
Affinity DataIC50: 0.760nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783851(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.760nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783870(N-(Cis-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-1-...)
Affinity DataIC50: 0.830nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783878(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.830nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM50382290(RGH-188 HCL | CARIPRAZINE HYDROCHLORIDE | US202402...)
Affinity DataIC50: 0.890nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783881(N-(4-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)e...)
Affinity DataIC50: 0.900nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783876(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.910nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783877(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 0.960nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783871(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 1.03nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783880(3-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 1.29nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783858(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 1.52nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783874(2-((Trans-4-(2-((R)-4-(benzo[b]thiophen-4-yl)-2-me...)
Affinity DataIC50: 1.58nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783854(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 1.59nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783867(1-(Cis-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-1-...)
Affinity DataIC50: 2.07nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783880(3-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 2.16nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783879(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 2.43nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783874(2-((Trans-4-(2-((R)-4-(benzo[b]thiophen-4-yl)-2-me...)
Affinity DataIC50: 2.59nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783868(3-(4-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)e...)
Affinity DataIC50: 2.69nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783851(N-(Trans-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-...)
Affinity DataIC50: 3.40nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783859(3-(Cis-4-(2-(4-(benzo[b]thiophen-4-yl)piperazin-1-...)
Affinity DataIC50: 4.25nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM783868(3-(4-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)e...)
Affinity DataIC50: 6.45nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandPNGBDBM50382290(RGH-188 HCL | CARIPRAZINE HYDROCHLORIDE | US202402...)
Affinity DataIC50: 191nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2026
Entry Details US Patent