Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 13437
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793471BDBM793471(US12559487, Example 6)
Affinity DataIC50: 2.70E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793481BDBM793481(US12559487, Example 17)
Affinity DataIC50: 3.00E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793479BDBM793479(US12559487, Example 14)
Affinity DataIC50: 3.20E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793483BDBM793483(US12559487, Example 19b)
Affinity DataIC50: 4.50E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793485BDBM793485(US12559487, Example 22)
Affinity DataIC50: 5.80E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793482BDBM793482(US12559487, Example 19a)
Affinity DataIC50: 6.00E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793492BDBM793492(US12559487, Example 30)
Affinity DataIC50: 7.30E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793487BDBM793487(US12559487, Example 25)
Affinity DataIC50: 9.70E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793473BDBM793473(US12559487, Example 8)
Affinity DataIC50: 9.70E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793480BDBM793480(US12559487, Example 15)
Affinity DataIC50: 1.70E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793468BDBM793468(US12559487, Example 3)
Affinity DataIC50: 1.80E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793470BDBM793470(US12559487, Example 5)
Affinity DataIC50: 2.10E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793478BDBM793478(US12559487, Example 13)
Affinity DataIC50: 2.60E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793466BDBM793466(2-(3-{1-[(3S)-2-Azabicyclo[2.2.2]octane-3-carbonyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793477BDBM793477(US12559487, Example 12)
Affinity DataIC50: 3.20E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793484BDBM793484(US12559487, Example 20)
Affinity DataIC50: 3.20E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793474BDBM793474(US12559487, Example 9)
Affinity DataIC50: 3.70E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793476BDBM793476(US12559487, Example 11)
Affinity DataIC50: 3.90E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793472BDBM793472(US12559487, Example 7)
Affinity DataIC50: 4.00E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793467BDBM793467(US12559487, Example 2)
Affinity DataIC50: 5.40E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793475BDBM793475(US12559487, Example 10)
Affinity DataIC50: 5.50E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793486BDBM793486(US12559487, Example 24)
Affinity DataIC50: 6.70E+4nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793469BDBM793469(US12559487, Example 4)
Affinity DataIC50: 1.00E+5nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793491BDBM793491(US12559487, Example 29)
Affinity DataIC50: 1.00E+5nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793490BDBM793490(US12559487, Example 28)
Affinity DataIC50: 1.00E+5nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793489BDBM793489(US12559487, Example 27)
Affinity DataIC50: 1.00E+5nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sumitomo Pharma Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 793488BDBM793488(US12559487, Example 26)
Affinity DataIC50: 1.00E+5nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
7/6/2026
Entry Details
US Patent