Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 13556
TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689197BDBM689197(US20240254109, Example 17A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 0.300nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689195BDBM689195(US20240254109, Example 15A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 0.310nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803699BDBM803699(US12617759, Example 24A)
Affinity DataIC50: 0.330nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803697BDBM803697(US12617759, Example 22A)
Affinity DataIC50: 0.340nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803690BDBM803690(US12617759, Example 20A)
Affinity DataIC50: 0.370nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689199BDBM689199(US20240254109, Example 19A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 0.400nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689198BDBM689198(US20240254109, Example 18A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 0.420nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689189BDBM689189(US20240254109, Example 7A | N-(Trans-3-(2-(4-(2,3-...)
Affinity DataIC50: 0.440nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689190BDBM689190(US20240254109, Example 11 | N-(3-(2-(4-(2,3-Dichlo...)
Affinity DataIC50: 0.620nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689187BDBM689187(US20240254109, Example 6A | N-(Trans-3-(2-(4-(2,3-...)
Affinity DataIC50: 0.75nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689203BDBM689203(US20240254109, Example 25 | N-(3-(2-(4-(2,3-Dichlo...)
Affinity DataIC50: 0.790nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689189BDBM689189(US20240254109, Example 7A | N-(Trans-3-(2-(4-(2,3-...)
Affinity DataIC50: 0.790nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 263449BDBM263449(US9550741, RGH-188 | US12617759, Example Cariprazi...)
Affinity DataIC50: 0.890nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689186BDBM689186(US20240254109, Example 4A | US12617759, Example 11...)
Affinity DataIC50: 0.950nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689195BDBM689195(US20240254109, Example 15A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 0.980nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689202BDBM689202(US20240254109, Example 24 | 3-(3-(2-(4-(Benzo[b]th...)
Affinity DataIC50: 1.13nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803697BDBM803697(US12617759, Example 22A)
Affinity DataIC50: 1.35nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689193BDBM689193(US20240254109, Example 13A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 1.36nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689198BDBM689198(US20240254109, Example 18A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 1.37nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803699BDBM803699(US12617759, Example 24A)
Affinity DataIC50: 1.80nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689193BDBM689193(US20240254109, Example 13A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 1.81nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689199BDBM689199(US20240254109, Example 19A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 1.89nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689197BDBM689197(US20240254109, Example 17A | N-(Trans-3-(2-(4-(2,3...)
Affinity DataIC50: 1.92nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689200BDBM689200(US20240254109, Example 20 | 1-Cyclopropyl-3-(3-(2-...)
Affinity DataIC50: 1.99nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803695BDBM803695(US12617759, Example 20B)
Affinity DataIC50: 2.54nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689201BDBM689201(US20240254109, Example 22 | (R) N-(3-(2-(4-(2,3-Di...)
Affinity DataIC50: 2.78nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803690BDBM803690(US12617759, Example 20A)
Affinity DataIC50: 4.19nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

TargetD(3) dopamine receptor(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689188BDBM689188(US20240254109, Example 6B | N-(Cis-3-(2-(4-(2,3-di...)
Affinity DataIC50: 4.37nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689187BDBM689187(US20240254109, Example 6A | N-(Trans-3-(2-(4-(2,3-...)
Affinity DataIC50: 5.77nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689203BDBM689203(US20240254109, Example 25 | N-(3-(2-(4-(2,3-Dichlo...)
Affinity DataIC50: 6.35nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689202BDBM689202(US20240254109, Example 24 | 3-(3-(2-(4-(Benzo[b]th...)
Affinity DataIC50: 6.39nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 803695BDBM803695(US12617759, Example 20B)
Affinity DataIC50: 8.73nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689201BDBM689201(US20240254109, Example 22 | (R) N-(3-(2-(4-(2,3-Di...)
Affinity DataIC50: 9.63nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689200BDBM689200(US20240254109, Example 20 | 1-Cyclopropyl-3-(3-(2-...)
Affinity DataIC50: 19.1nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689186BDBM689186(US20240254109, Example 4A | US12617759, Example 11...)
Affinity DataIC50: 41.5nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689190BDBM689190(US20240254109, Example 11 | N-(3-(2-(4-(2,3-Dichlo...)
Affinity DataIC50: 44nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 689188BDBM689188(US20240254109, Example 6B | N-(Cis-3-(2-(4-(2,3-di...)
Affinity DataIC50: 48.5nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Hansoh Biomedical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 263449BDBM263449(US9550741, RGH-188 | US12617759, Example Cariprazi...)
Affinity DataIC50: 191nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2026
Entry Details
US Patent