Compile Data Set for Download or QSAR
Report error Found 552 Enz. Inhib. hit(s) with all data for entry = 13593
TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809293BDBM809293((Z)-2-(benzo[d]thiazol-6-yl(2-methoxyethyl)amino)-...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809267BDBM809267((Z)-5-(benzo[d]thiazol-5-ylmethylene)-2-(benzo[d]t...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809267BDBM809267((Z)-5-(benzo[d]thiazol-5-ylmethylene)-2-(benzo[d]t...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1 [156-555](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809267BDBM809267((Z)-5-(benzo[d]thiazol-5-ylmethylene)-2-(benzo[d]t...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809292BDBM809292((Z)-2-(benzo[d]thiazol-6-ylamino)-5-(benzo[d]thiaz...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809292BDBM809292((Z)-2-(benzo[d]thiazol-6-ylamino)-5-(benzo[d]thiaz...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809265BDBM809265((Z)-5-((1H-indazol-5-yl)methylene)-2-(phenylamino)...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809244BDBM809244((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((cyclopro...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809266BDBM809266((4Z)-4-[(1H-1,2,3-benzotriazol-6-yl)methylidene]-2...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809266BDBM809266((4Z)-4-[(1H-1,2,3-benzotriazol-6-yl)methylidene]-2...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809265BDBM809265((Z)-5-((1H-indazol-5-yl)methylene)-2-(phenylamino)...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809273BDBM809273((Z)-2-((1H-indol-5-yl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809297BDBM809297((Z)-5-(benzo[d]thiazol-6-ylmethylene)-24(1-methyl-...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809251BDBM809251((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-(benzyl(ph...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 2 [1-640](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809273BDBM809273((Z)-2-((1H-indol-5-yl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK2 (1 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809297BDBM809297((Z)-5-(benzo[d]thiazol-6-ylmethylene)-24(1-methyl-...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809274BDBM809274((Z)-5-(benzo[d][1,3]dioxol-5-ylmethylene)-2-(benzo...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809226BDBM809226((4Z)-2-(phenylamino)-4-[(quinoxalin-6-yl)methylide...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809295BDBM809295(N-(1,3-benzothiazol-6-yl)-N-[(4Z)-4-[(1,3-benzothi...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809226BDBM809226((4Z)-2-(phenylamino)-4-[(quinoxalin-6-yl)methylide...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 2 [1-640](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809295BDBM809295(N-(1,3-benzothiazol-6-yl)-N-[(4Z)-4-[(1,3-benzothi...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK2 (1 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809250BDBM809250((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((4-chloro...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809296BDBM809296((Z)-2-(benzo[d]thiazol-6-ylamino)-5-(thiazol-5-ylm...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809273BDBM809273((Z)-2-((1H-indol-5-yl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809294BDBM809294((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((2-methyl...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809294BDBM809294((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((2-methyl...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 2 [1-640](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809294BDBM809294((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((2-methyl...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK2 (1 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha'(Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809294BDBM809294((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((2-methyl...)
Affinity DataIC50: 100nMAssay Description:Briefly, CK2a2 (CSNK2a2) (7 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809271BDBM809271((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((1-methyl...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809295BDBM809295(N-(1,3-benzothiazol-6-yl)-N-[(4Z)-4-[(1,3-benzothi...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809281BDBM809281((Z)-5-((1-methyl-1H-indazol-5-yl)methylene)-2-(phe...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809235BDBM809235((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((4-methox...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809305BDBM809305((Z)-2-(benzo[b]thiophen-5-ylamino)-5-(benzo[d]thia...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809235BDBM809235((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-((4-methox...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809258BDBM809258((Z)-2-(benzo[d]thiazol-6-ylamino)-5-(benzo[d]thiaz...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809258BDBM809258((Z)-2-(benzo[d]thiazol-6-ylamino)-5-(benzo[d]thiaz...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809256BDBM809256((Z)-5-((1-methyl-1H-benzo[d]imidazol-6-yl)methylen...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809279BDBM809279((Z)-2-(benzo[d]thiazol-6-ylamino)-5-((1-methyl-1H-...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809256BDBM809256((Z)-5-((1-methyl-1H-benzo[d]imidazol-6-yl)methylen...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 1 [156-555](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809279BDBM809279((Z)-2-(benzo[d]thiazol-6-ylamino)-5-((1-methyl-1H-...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK1 (4 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 2 [1-640](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809279BDBM809279((Z)-2-(benzo[d]thiazol-6-ylamino)-5-((1-methyl-1H-...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK2 (1 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809303BDBM809303((Z)-2-(benzo[d]thiazol-6-yl(benzyl)amino)-5-(benzo...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha'(Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809256BDBM809256((Z)-5-((1-methyl-1H-benzo[d]imidazol-6-yl)methylen...)
Affinity DataIC50: 100nMAssay Description:Briefly, CK2a2 (CSNK2a2) (7 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809280BDBM809280((Z)-5-((1H-benzo[d]imidazol-6-yl)methylene)-2-(ben...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809280BDBM809280((Z)-5-((1H-benzo[d]imidazol-6-yl)methylene)-2-(ben...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 2 [1-640](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809301BDBM809301((Z)-2-((1H-benzo[d]imidazol-6-yl)amino)-5-(benzo[d...)
Affinity DataIC50: 100nMAssay Description:Briefly, HIPK2 (1 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809255BDBM809255((Z)-5-(benzo[d]thiazol-6-ylmethylene)-2-(isopropyl...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 809302BDBM809302((Z)-2-((4-aminophenyl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 100nMAssay Description:Briefly, DYRK1A (3 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentr...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809302BDBM809302((Z)-2-((4-aminophenyl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 100nMAssay Description:Briefly, CLK1 (16 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various concentra...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

TargetCasein kinase II subunit alpha'(Human)
Tongji University

US Patent
LigandChemical structure of BindingDB Monomer ID 809302BDBM809302((Z)-2-((4-aminophenyl)amino)-5-(benzo[d]thiazol-6-...)
Affinity DataIC50: 100nMAssay Description:Briefly, CK2a2 (CSNK2a2) (7 nM) in the enzymatic buffer solutions (40 mM Tris, pH 7.5, 20 mM MgCl2, 0.1 mg/ml BSA, 50 μM DTT) were mixed with various...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/19/2026
Entry Details
US Patent

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