Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 11458
TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617530BDBM617530(US20230286925, Compound HYBI_087)
Affinity DataIC50: 2.60nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617532BDBM617532(US20230286925, Compound HYBI_110)
Affinity DataIC50: 3nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617525BDBM617525(US20230286925, Compound HYBI_083)
Affinity DataIC50: 3.08nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617531BDBM617531(US20230286925, Compound HYBI_101)
Affinity DataIC50: 3.65nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617528BDBM617528(US20230286925, Compound HYBI_085)
Affinity DataIC50: 3.86nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617529BDBM617529(US20230286925, Compound HYBI_086)
Affinity DataIC50: 3.99nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617526BDBM617526(US20230286925, Compound HYBI_084)
Affinity DataIC50: 4.72nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617524BDBM617524(US20230286925, Compound HYBI_082)
Affinity DataIC50: 4.91nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617511BDBM617511(US20230286925, Compound HYBI_028)
Affinity DataIC50: 5.24nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617507BDBM617507(US20230286925, Compound HYBI_021)
Affinity DataIC50: 7.09nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617506BDBM617506(US20230286925, Compound HYBI_020)
Affinity DataIC50: 8.23nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617500BDBM617500(US20230286925, Compound HYBI_010)
Affinity DataIC50: 9.62nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617510BDBM617510(US20230286925, Compound HYBI_027)
Affinity DataIC50: 10.8nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617499BDBM617499(US20230286925, Compound HYBI_003)
Affinity DataIC50: 15.6nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617503BDBM617503(US20230286925, Compound HYBI_018)
Affinity DataIC50: 16.8nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617505BDBM617505(US20230286925, Compound HYBI_019A)
Affinity DataIC50: 17.1nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617501BDBM617501(US20230286925, Compound HYBI_013)
Affinity DataIC50: 19.4nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617523BDBM617523(US20230286925, Compound HYBI_053)
Affinity DataIC50: 19.4nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617509BDBM617509(US20230286925, Compound HYBI_023)
Affinity DataIC50: 19.8nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617504BDBM617504(US20230286925, Compound HYBI_019)
Affinity DataIC50: 20.4nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617502BDBM617502(US20230286925, Compound HYBI_016)
Affinity DataIC50: 20.6nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617497BDBM617497(US20230286925, Compound HYBI_002)
Affinity DataIC50: 44.2nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617508BDBM617508(US20230286925, Compound HYBI_022)
Affinity DataIC50: 62.3nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617512BDBM617512(US20230286925, Compound HYBI_037)
Affinity DataIC50: 109nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617514BDBM617514(US20230286925, Compound HYBI_039)
Affinity DataIC50: 131nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617513BDBM617513(US20230286925, Compound HYBI_038)
Affinity DataIC50: 185nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617520BDBM617520(US20230286925, Compound HYBI_046)
Affinity DataIC50: 271nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617519BDBM617519(US20230286925, Compound HYBI_045)
Affinity DataIC50: 384nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617521BDBM617521(US20230286925, Compound HYBI_047)
Affinity DataIC50: 466nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617516BDBM617516(US20230286925, Compound HYBI_042)
Affinity DataIC50: 802nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617515BDBM617515(US20230286925, Compound HYBI_040)
Affinity DataIC50: 828nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617518BDBM617518(US20230286925, Compound HYBI_044)
Affinity DataIC50: 903nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandChemical structure of BindingDB Monomer ID 617522BDBM617522(US20230286925, Compound HYBI_050)
Affinity DataIC50: 5.56E+3nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent