Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 11458
TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617530(US20230286925, Compound HYBI_087)
Affinity DataIC50: 2.60nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617532(US20230286925, Compound HYBI_110)
Affinity DataIC50: 3nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617525(US20230286925, Compound HYBI_083)
Affinity DataIC50: 3.08nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617531(US20230286925, Compound HYBI_101)
Affinity DataIC50: 3.65nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617528(US20230286925, Compound HYBI_085)
Affinity DataIC50: 3.86nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617529(US20230286925, Compound HYBI_086)
Affinity DataIC50: 3.99nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617526(US20230286925, Compound HYBI_084)
Affinity DataIC50: 4.72nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617524(US20230286925, Compound HYBI_082)
Affinity DataIC50: 4.91nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617511(US20230286925, Compound HYBI_028)
Affinity DataIC50: 5.24nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617507(US20230286925, Compound HYBI_021)
Affinity DataIC50: 7.09nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617506(US20230286925, Compound HYBI_020)
Affinity DataIC50: 8.23nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617500(US20230286925, Compound HYBI_010)
Affinity DataIC50: 9.62nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617510(US20230286925, Compound HYBI_027)
Affinity DataIC50: 10.8nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617499(US20230286925, Compound HYBI_003)
Affinity DataIC50: 15.6nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617503(US20230286925, Compound HYBI_018)
Affinity DataIC50: 16.8nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617505(US20230286925, Compound HYBI_019A)
Affinity DataIC50: 17.1nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617501(US20230286925, Compound HYBI_013)
Affinity DataIC50: 19.4nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617523(US20230286925, Compound HYBI_053)
Affinity DataIC50: 19.4nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617509(US20230286925, Compound HYBI_023)
Affinity DataIC50: 19.8nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617504(US20230286925, Compound HYBI_019)
Affinity DataIC50: 20.4nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617502(US20230286925, Compound HYBI_016)
Affinity DataIC50: 20.6nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617497(US20230286925, Compound HYBI_002)
Affinity DataIC50: 44.2nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617508(US20230286925, Compound HYBI_022)
Affinity DataIC50: 62.3nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617512(US20230286925, Compound HYBI_037)
Affinity DataIC50: 109nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617514(US20230286925, Compound HYBI_039)
Affinity DataIC50: 131nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617513(US20230286925, Compound HYBI_038)
Affinity DataIC50: 185nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617520(US20230286925, Compound HYBI_046)
Affinity DataIC50: 271nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617519(US20230286925, Compound HYBI_045)
Affinity DataIC50: 384nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617521(US20230286925, Compound HYBI_047)
Affinity DataIC50: 466nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617516(US20230286925, Compound HYBI_042)
Affinity DataIC50: 802nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617515(US20230286925, Compound HYBI_040)
Affinity DataIC50: 828nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617518(US20230286925, Compound HYBI_044)
Affinity DataIC50: 903nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent

TargetHistone-lysine N-methyltransferase 2A(Human)
Huyabio International

US Patent
LigandPNGBDBM617522(US20230286925, Compound HYBI_050)
Affinity DataIC50: 5.56E+3nMAssay Description:WDR5 TR-FRET Assay Procedure: Stock compounds were transferred to the assay plate by Echo Liquid Handler. Reactions were performed in the assay buffe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2023
Entry Details
US Patent