Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 11482
TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620107BDBM620107((R)-3-methyl-4-(8-(1-methyl-1H-pyrazol-5-yl)-3-(1H...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620108BDBM620108((R)-3-methyl-4-(8-(1-(methylsulfonyl)cyclopropyl)-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620109BDBM620109((R)-3-methyl-4-(4-(1-methyl-1H-pyrazol-5-yl)-7-(1H...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620110BDBM620110((R)-3-methyl-4-(7-(1-methyl-1H-pyrazol-5-yl)-3-(1H...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620103BDBM620103((R)-4-(3,7-di(1H-pyrazol-5-yl)pyrazolo[1,5-a]pyrim...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620104BDBM620104((R)-3-methyl-4-(3-(3-methyl-1H-pyrazol-5-yl)-7-(1-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620106BDBM620106((R)-3-methyl-4-(7-(1-methyl-1H-pyrazol-5-yl)-3-(3-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620115BDBM620115((R)-3-methyl-4-(4-(1-methyl-1H-pyrazol-5-yl)-7-(3-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620116BDBM620116((3R)-4-[4-(diethylphosphoryl)-7-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620117BDBM620117((R)-4-(7-(1,4-dimethyl-1H-1,2,3-triazol-5-yl)-3-(3...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620118BDBM620118((R)-3-methyl-4-(3-(3-methyl-1H-pyrazol-5-yl)-7-(1-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620111BDBM620111((R)-3-methyl-4-(4-(1-(methylsulfonyl)cyclopropyl)-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620112BDBM620112((R)-3-methyl-4-(7-(3-methyl-1H-pyrazol-5-yl)-4-(1-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620113BDBM620113((1R,5S)-3-(4-(1-(methylsulfonyl)cyclopropyl)-7-(1H...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620114BDBM620114((3R)-4-[4-(dimethyl-1H-1,2,3-triazol-5-yl)-7-(1H-p...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620093BDBM620093((R)-3-methyl-4-(7-(1-methyl-1H-pyrazol-5-yl)-3-(1H...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620099BDBM620099((R)-imino(methyl)(1-(5-((R)-3-methylmorpholino)-3-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620100BDBM620100((S)-imino(methyl)(1-(5-((R)-3-methylmorpholino)-3-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620101BDBM620101((R)-3-methyl-4-(7-(1-(methylsulfonyl)cyclopropyl)-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620102BDBM620102((R)-3-methyl-4-(7-(1-(methylsulfonyl)cyclopropyl)-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620096BDBM620096((R)-3-methyl-4-(7-(1-methyl-1H-pyrazol-5-yl)-3-(1H...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620097BDBM620097((R)-3-methyl-4-(7-(1-(methylsulfonyl)cyclopropyl)-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620098BDBM620098((R)-4-(7-(2-fluoropyridin-3-yl)-3-(1H-pyrazol-5-yl...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620139BDBM620139((R)-1-(3-(3-methyl-1H-pyrazol-5-yl)-5-(3-methylmor...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620140BDBM620140((R)-1-(5-(3-methylmorpholino)-3-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620135BDBM620135(US20230295166, Compound 82)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620136BDBM620136((R)-4-(5-(3-methylmorpholino)-3-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620137BDBM620137((R)-4-(3-(3-methyl-1H-pyrazol-5-yl)-5-(3-methylmor...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620138BDBM620138((R)-4-(7-(cyclopropylsulfonyl)-3-(3-methyl-1H-pyra...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620123BDBM620123((R)-3-methyl-4-(3-(3-methyl-1H-pyrazol-5-yl)-7-(2-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620124BDBM620124((R)-1-(5-(3-methylmorpholino)-3-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620125BDBM620125((R)-1-(5-(3-methylmorpholino)-3-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620126BDBM620126((R)-1-(2-(3-methylmorpholino)-7-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620119BDBM620119((R)-1-(5-(3-methylmorpholino)-3-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620120BDBM620120((R)-1-(3-(3-methyl-1H-pyrazol-5-yl)-5-(3-methylmor...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620119BDBM620119((R)-1-(5-(3-methylmorpholino)-3-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620122BDBM620122((R)-3-methyl-4-(7-(2-(methylsulfony])propan-2-yl)-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620131BDBM620131((R)-4-(7-(cyclopropylsulfonyl)-3-(1H-pyrazol-5-yl)...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620132BDBM620132((R)-2-(5-(3-methylmorpholino)-3-(1H-pyrazol-5-yl)i...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620133BDBM620133((R)-1-(3-(3-methyl-1H-pyrazol-5-yl)-5-(3-methylmor...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620134BDBM620134((R)-1-(3-(3-methyl-1H-pyrazol-5-yl)-5-(3-methylmor...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620127BDBM620127((3R)-4-[5-chloro-4-(1-methyl-1H-pyrazol-5-yl)-7-(1...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620128BDBM620128((R)-4-(5-chloro-4-(1-methyl-1H-pyrazol-5-yl)-7-(3-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620129BDBM620129((R)-1-(7-(3-methyl-1H-pyrazol-5-yl)-2-(3-methylmor...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620130BDBM620130((R)-2-methyl-2-(7-(3-methyl-1H-pyrazol-5-yl)-2-(3-...)
Affinity DataIC50: 100nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620095BDBM620095((R)-3-methyl-4-(7-(1-methyl-1H-pyrazol-5-yl)-3-(py...)
Affinity DataIC50: 300nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620094BDBM620094((R)-3-methyl-4-(7-(1-methyl-1H-pyrazol-5-yl)-3-(1H...)
Affinity DataIC50: 500nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Antengene Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 620105BDBM620105((R)-3-methyl-4-(3-(4-methyl-1H-pyrazol-5-yl)-7-(1-...)
Affinity DataIC50: 500nMAssay Description:Detection of ATR kinase activity utilized the Mobility shift assay to measure the phosphorylation of the substrate protein FAM-RAD17 (GL, Cat. No. 51...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent