Compile Data Set for Download or QSAR
Report error Found 176 Enz. Inhib. hit(s) with all data for entry = 12142
TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609784BDBM609784(US11707539, Compound 6591 | US20240207292, Compoun...)
Affinity DataIC50: 0.360nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682328BDBM682328(US20240207292, Compound 6590LU)
Affinity DataIC50: 0.400nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609722BDBM609722(US11707539, Compound 6555 | DOTA- aminomethyl-Bz- ...)
Affinity DataIC50: 0.700nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609430BDBM609430(US11707539, Compound 6489 | DOTA[Cu(II)]- GABA-HyB...)
Affinity DataIC50: 0.800nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609427BDBM609427(US11707539, Compound 6489S | DOTA-GABA- HyBz-D-Ala...)
Affinity DataIC50: 0.800nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609787BDBM609787(US11707539, Compound 6958LU | US20240207292, Compo...)
Affinity DataIC50: 1nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682244BDBM682244(US20240207292, Compound 2054 | Val-boroPro)
Affinity DataIC50: 1nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682325BDBM682325(US20240207292, Compound 6489-GD)
Affinity DataIC50: 1.10nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682270BDBM682270(US20240207292, Compound 6489Gd | DOTA[Gd]- GABA-Hy...)
Affinity DataIC50: 1.10nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682332BDBM682332(US20240207292, Compound 6958LU)
Affinity DataIC50: 1.10nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609755BDBM609755(US11707539, Compound 6869 | US20240207292, Compoun...)
Affinity DataIC50: 1.10nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609781BDBM609781(US11707539, Compound 6590 | US20240207292, Compoun...)
Affinity DataIC50: 1.60nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609535BDBM609535(US11707539, Compound 6572 | DOTA-PABA-D- Ala-boroP...)
Affinity DataIC50: 1.60nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609535BDBM609535(US11707539, Compound 6572 | DOTA-PABA-D- Ala-boroP...)
Affinity DataIC50: 1.60nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609441BDBM609441(US11707539, Compound 6486S | DOTA-EACA- HyBz-D-Ala...)
Affinity DataIC50: 1.70nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682338BDBM682338(US20240207292, Compound 4613-C)
Affinity DataIC50: 1.70nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609721BDBM609721(US11707539, Compound 6551 | Lys(GABA- DOTA)-boroPr...)
Affinity DataIC50: 2nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609414BDBM609414(US11707539, Compound 6487S | DOTA-Gly- HyBz-D-Ala-...)
Affinity DataIC50: 2.10nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609417BDBM609417(DOTA[Cu(II)]- Gly-HyBz-D-Ala- boroPro | BDBM609769...)
Affinity DataIC50: 2.10nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609723BDBM609723(US11707539, Compound 6556 | DOTA- aminomethyl-Nic-...)
Affinity DataIC50: 2.40nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609723BDBM609723(US11707539, Compound 6556 | DOTA- aminomethyl-Nic-...)
Affinity DataIC50: 2.40nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609430BDBM609430(US11707539, Compound 6489 | DOTA[Cu(II)]- GABA-HyB...)
Affinity DataIC50: 2.60nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609721BDBM609721(US11707539, Compound 6551 | Lys(GABA- DOTA)-boroPr...)
Affinity DataIC50: 2.60nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609379BDBM609379(US11707539, Compound 4536B | DOTA-HyBz-D- Ala-boro...)
Affinity DataIC50: 2.70nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609481BDBM609481(US11707539, Compound 6486 | DOTA[Cu(II)]- EACA-HyB...)
Affinity DataIC50: 2.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609481BDBM609481(US11707539, Compound 6486 | DOTA[Cu(II)]- EACA-HyB...)
Affinity DataIC50: 2.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609718BDBM609718(US11707539, Compound 6549 | Lys(DOTA)- boroPro | U...)
Affinity DataIC50: 2.90nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609775BDBM609775(US11707539, Compound 6556LU | US20240207292, Compo...)
Affinity DataIC50: 2.90nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609718BDBM609718(US11707539, Compound 6549 | Lys(DOTA)- boroPro | U...)
Affinity DataIC50: 3.20nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609786BDBM609786(US11707539, Compound 6958 | US20240207292, Compoun...)
Affinity DataIC50: 3.20nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609719BDBM609719(DOTA-Gly-Gly- Val-D-Ala- boroPro | US11707539, Com...)
Affinity DataIC50: 3.5nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609720BDBM609720(US11707539, Compound 6522CU | DOTA[(Cu(II)]- Gly-G...)
Affinity DataIC50: 3.5nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609722BDBM609722(US11707539, Compound 6555 | DOTA- aminomethyl-Bz- ...)
Affinity DataIC50: 3.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609788BDBM609788(US11707539, Compound 6952 | US20240207292, Compoun...)
Affinity DataIC50: 4.70nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609759BDBM609759(US11707539, Compound 6940 | US20240207292, Compoun...)
Affinity DataIC50: 5.20nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682273BDBM682273(US20240207292, Compound 5183 | DOTA[(Gd(III)]- HyB...)
Affinity DataIC50: 5.30nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682244BDBM682244(US20240207292, Compound 2054 | Val-boroPro)
Affinity DataIC50: 5.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609717BDBM609717(US11707539, Compound 6521 | DOTA-Gly-Val- D-Ala-bo...)
Affinity DataIC50: 6.90nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609717BDBM609717(US11707539, Compound 6521 | DOTA-Gly-Val- D-Ala-bo...)
Affinity DataIC50: 6.90nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682279BDBM682279(US20240207292, Compound 6522L)
Affinity DataIC50: 7.60nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609720BDBM609720(US11707539, Compound 6522CU | DOTA[(Cu(II)]- Gly-G...)
Affinity DataIC50: 8.70nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609771BDBM609771(US11707539, Compound 6487LU | US20240207292, Compo...)
Affinity DataIC50: 8.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609419BDBM609419(US11707539, Compound 6488S | DOTA-betaAla- HyBz-D-...)
Affinity DataIC50: 8.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 682337BDBM682337(US20240207292, Compound 4613-B)
Affinity DataIC50: 8.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609417BDBM609417(DOTA[Cu(II)]- Gly-HyBz-D-Ala- boroPro | BDBM609769...)
Affinity DataIC50: 8.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609419BDBM609419(US11707539, Compound 6488S | DOTA-betaAla- HyBz-D-...)
Affinity DataIC50: 8.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609417BDBM609417(DOTA[Cu(II)]- Gly-HyBz-D-Ala- boroPro | BDBM609769...)
Affinity DataIC50: 8.80nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609740BDBM609740(US11707539, Compound 6795 | US20240207292, Compoun...)
Affinity DataIC50: 8.90nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609765BDBM609765(US11707539, Compound 4536 | US20240207292, Compoun...)
Affinity DataIC50: 9nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandChemical structure of BindingDB Monomer ID 609756BDBM609756(US11707539, Compound 6870 | US20240207292, Compoun...)
Affinity DataIC50: 9.20nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

Displayed 1 to 50 (of 176 total ) | Next | Last >>
Jump to: