Compile Data Set for Download or QSAR
Report error Found 338 Enz. Inhib. hit(s) with all data for entry = 12433
LigandChemical structure of BindingDB Monomer ID 702242BDBM702242(US20240360137, Example 41)
Affinity DataIC50: 5nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702270BDBM702270(US20240360137, Example 69)
Affinity DataIC50: 6nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702282BDBM702282(US20240360137, Example 81)
Affinity DataIC50: 6nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702233BDBM702233(US20240360137, Example 32)
Affinity DataIC50: 6nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702271BDBM702271(US20240360137, Example 70)
Affinity DataIC50: 6nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702269BDBM702269(US20240360137, Example 68)
Affinity DataIC50: 7nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702240BDBM702240(US20240360137, Example 39)
Affinity DataIC50: 7nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702204BDBM702204(US20240360137, Example 3)
Affinity DataIC50: 7nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702221BDBM702221(US20240360137, Example 20)
Affinity DataIC50: 8nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702239BDBM702239(US20240360137, Example 38)
Affinity DataIC50: 8nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702257BDBM702257(US20240360137, Example 56)
Affinity DataIC50: 10nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702235BDBM702235(US20240360137, Example 34)
Affinity DataIC50: 10nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702246BDBM702246(US20240360137, Example 45)
Affinity DataIC50: 11nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702229BDBM702229(US20240360137, Example 28)
Affinity DataIC50: 11nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702228BDBM702228(US20240360137, Example 27)
Affinity DataIC50: 11nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702256BDBM702256(US20240360137, Example 55)
Affinity DataIC50: 11nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702214BDBM702214(US20240360137, Example 13)
Affinity DataIC50: 12nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702225BDBM702225(US20240360137, Example 24)
Affinity DataIC50: 12nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702265BDBM702265(US20240360137, Example 64)
Affinity DataIC50: 12nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702250BDBM702250(US20240360137, Example 49)
Affinity DataIC50: 15nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702258BDBM702258(US20240360137, Example 57)
Affinity DataIC50: 15nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702245BDBM702245(US20240360137, Example 44)
Affinity DataIC50: 15nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702224BDBM702224(US20240360137, Example 23)
Affinity DataIC50: 15nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702259BDBM702259(US20240360137, Example 58)
Affinity DataIC50: 16nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702222BDBM702222(US20240360137, Example 21)
Affinity DataIC50: 17nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702263BDBM702263(US20240360137, Example 62)
Affinity DataIC50: 17nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702279BDBM702279(US20240360137, Example 78)
Affinity DataIC50: 17nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702203BDBM702203(Synthesis of | US20240360137, Example 2)
Affinity DataIC50: 18nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702244BDBM702244(US20240360137, Example 43)
Affinity DataIC50: 19nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702213BDBM702213(US20240360137, Example 12)
Affinity DataIC50: 20nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702232BDBM702232(US20240360137, Example 31)
Affinity DataIC50: 21nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702249BDBM702249(US20240360137, Example 48)
Affinity DataIC50: 22nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702231BDBM702231(US20240360137, Example 30)
Affinity DataIC50: 22nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702268BDBM702268(US20240360137, Example 67)
Affinity DataIC50: 23nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702226BDBM702226(US20240360137, Example 25)
Affinity DataIC50: 24nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702243BDBM702243(US20240360137, Example 42)
Affinity DataIC50: 24nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702230BDBM702230(US20240360137, Example 29)
Affinity DataIC50: 26nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702241BDBM702241(US20240360137, Example 40)
Affinity DataIC50: 26nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702283BDBM702283(US20240360137, Example 82)
Affinity DataIC50: 26nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702286BDBM702286(US20240360137, Example 85)
Affinity DataIC50: 27nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702248BDBM702248(US20240360137, Example 47)
Affinity DataIC50: 27nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702281BDBM702281(US20240360137, Example 80)
Affinity DataIC50: 29nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702215BDBM702215(US20240360137, Example 14)
Affinity DataIC50: 30nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702238BDBM702238(US20240360137, Example 37)
Affinity DataIC50: 31nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702253BDBM702253(US20240360137, Example 52)
Affinity DataIC50: 31nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702284BDBM702284(US20240360137, Example 83)
Affinity DataIC50: 31nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702277BDBM702277(US20240360137, Example 76)
Affinity DataIC50: 32nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702207BDBM702207(US20240360137, Example 6)
Affinity DataIC50: 32nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702223BDBM702223(US20240360137, Example 22)
Affinity DataIC50: 34nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 702202BDBM702202(Synthesis of | US20240360137, Example 1)
Affinity DataIC50: 38nMAssay Description:Biochemical assays measured the inhibitory effects of compounds in this disclosure on the enzymatic activity of CDK enzyme in complex with Cyclin pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2025
Entry Details
US Patent

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