Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 12441
TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702970BDBM702970(US20240366606, Compound 9-(ZINC49534341))
Affinity DataKi:  32nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702976BDBM702976(US20240366606, Compound C9-6)
Affinity DataKi:  38nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702979BDBM702979(US20240366606, Compound C9-9)
Affinity DataKi:  47nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702964BDBM702964(US20240366606, Compound 1-(ZINC98174789))
Affinity DataKi:  57nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702969BDBM702969(US20240366606, Compound 8-(Z4655335085))
Affinity DataKi:  57nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 114420BDBM114420(3-[(2-methoxyphenyl)methyl]-2-sulfanylidene-1H-qui...)
Affinity DataKi:  98nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702972BDBM702972(US20240366606, Compound C9-1)
Affinity DataKi:  172nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702967BDBM702967(US20240366606, Compound 6-(ZINC71274619))
Affinity DataKi:  318nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702978BDBM702978(US20240366606, Compound C9-8)
Affinity DataKi:  514nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702966BDBM702966(US20240366606, Compound 5-(ZINC93327152))
Affinity DataKi:  895nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702977BDBM702977(US20240366606, Compound C9-7)
Affinity DataKi:  929nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702974BDBM702974(US20240366606, Compound C9-4)
Affinity DataKi:  1.17E+3nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702973BDBM702973(US20240366606, Compound C9-3)
Affinity DataKi:  1.78E+3nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702963BDBM702963(US20240366606, Compound ZINC16991592)
Affinity DataKi:  2.19E+3nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702971BDBM702971(US20240366606, Compound 14-(ZINC425284))
Affinity DataKi:  2.52E+3nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702965BDBM702965(US20240366606, Compound 2-(ZINC5286526))
Affinity DataKi:  6.18E+3nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetMas-related G-protein coupled receptor member X2(Human)
University of California

US Patent
LigandChemical structure of BindingDB Monomer ID 702968BDBM702968(US20240366606, Compound 7-(ZINC7045547))
Affinity DataKi:  6.52E+3nMAssay Description:HEK293 cells were cultured in DMEM with 4.5 g L-1 glucose, L-glutamine, and sodium pyruvate (Mediatech) containing 10% (v/v) FBS (Axenia BioLogix) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent