Compile Data Set for Download or QSAR
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 12445
TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703019BDBM703019(2-((5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro- l...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703018BDBM703018(2-((5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro- l...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703017BDBM703017(2-((5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro- l...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703016BDBM703016(2-((5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro- l...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703048BDBM703048(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703039BDBM703039(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703022BDBM703022(2-((5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro- l...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703037BDBM703037(US20240368078, Compound 54)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703026BDBM703026(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703025BDBM703025(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703047BDBM703047(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703030BDBM703030(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703046BDBM703046(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703061BDBM703061(2-cyclopropyl-2- ((3S,5R)-5-(2,3- dichloro-6- hydr...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703060BDBM703060(US20240368078, Compound 77)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703028BDBM703028(US20240368078, Compound 45)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703044BDBM703044(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 100nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703035BDBM703035(US20240368078, Compound 52)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703034BDBM703034(US20240368078, Compound 51)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703033BDBM703033(US20240368078, Compound 50)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703032BDBM703032(N-(((3R,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrr...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703038BDBM703038(2-((2R,4S)-4-((1H- pyrazol-3- yl)methyl)pyrrolidin...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703036BDBM703036(US20240368078, Compound 53)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703059BDBM703059(US20240368078, Compound 76)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703027BDBM703027(US20240368078, Compound 44)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703058BDBM703058(US20240368078, Compound 75)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703057BDBM703057(US20240368078, Compound 74)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703056BDBM703056(2-((3R,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703024BDBM703024(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703031BDBM703031(US20240368078, Compound 48)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703062BDBM703062(2-cyclopropyl-2- ((3S,5R)-5-(2,3- dichloro-6- hydr...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703029BDBM703029(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703051BDBM703051(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703050BDBM703050(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703049BDBM703049(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703023BDBM703023(2-((5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro- l...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703055BDBM703055(2-((3R,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703054BDBM703054(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703021BDBM703021(2-((5R)-5-(4,5- dichloro-2- hydroxyphenyl)pyrro- l...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703053BDBM703053(1-(3,3- bis(hydroxymethyl) azetidin-1-yl)-2- ((3S,...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703020BDBM703020(2-((5R)-5-(2,3- dichloro-6- hdyroxyphenyl)pyrro- l...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703052BDBM703052(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703043BDBM703043(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703042BDBM703042(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703041BDBM703041(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703040BDBM703040(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703015BDBM703015(US20240368078, Compound 32)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703014BDBM703014(US20240368078, Compound 31)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily A member 3(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703045BDBM703045(2-((3S,5R)-5-(2,3- dichloro-6- hydroxyphenyl)pyrro...)
Affinity DataIC50: 1.00E+3nMAssay Description:This assay is used to evaluate the disclosed compounds' activities as Kv1.3 potassium channel blockers. The cells were bathed in an extracellular...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
D.E. Shaw Research

US Patent
LigandChemical structure of BindingDB Monomer ID 703034BDBM703034(US20240368078, Compound 51)
Affinity DataIC50: 2.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
US Patent

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