Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 12464
LigandChemical structure of BindingDB Monomer ID 529296BDBM529296(US11198695, Example II-233 | US20240374587, Exampl...)
Affinity DataIC50: 0.220nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704328BDBM704328(US20240374587, Example I'-033 | US12227509, Exampl...)
Affinity DataIC50: 0.730nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704331BDBM704331(US20240374587, Example I'-066 | US12227509, Exampl...)
Affinity DataIC50: 0.850nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529357BDBM529357(US11198695, Example II-295 | US20240374587, Exampl...)
Affinity DataIC50: 1nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704332BDBM704332(US20240374587, Example I'-079 | US12227509, Exampl...)
Affinity DataIC50: 1.13nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529288BDBM529288(US11198695, Example II-225 | US20240374587, Exampl...)
Affinity DataIC50: 1.14nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704329BDBM704329(US20240374587, Example I'-046 | US12227509, Exampl...)
Affinity DataIC50: 1.17nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529160BDBM529160(US11198695, Example II-93 | US20240374587, Example...)
Affinity DataIC50: 1.21nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704337BDBM704337(US20240374587, Example I'-133 | US12227509, Exampl...)
Affinity DataIC50: 1.39nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529041BDBM529041(US11198695, Example I-253 | US20240374587, Example...)
Affinity DataIC50: 1.40nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704339BDBM704339(US20240374587, Example I'-137 | US12227509, Exampl...)
Affinity DataIC50: 1.53nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704335BDBM704335(US20240374587, Example I'-126 | US12227509, Exampl...)
Affinity DataIC50: 1.59nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529170BDBM529170(US11198695, Example II-103 | US20240374587, Exampl...)
Affinity DataIC50: 1.61nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704320BDBM704320(US20240374587, Example II-168)
Affinity DataIC50: 1.88nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704327BDBM704327(US20240374587, Example I'-020 | US12227509, Exampl...)
Affinity DataIC50: 1.97nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529063BDBM529063(US11198695, Example I-275 | US20240374587, Example...)
Affinity DataIC50: 2nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529217BDBM529217(US11198695, Example II-151 | US20240374587, Exampl...)
Affinity DataIC50: 2.05nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529238BDBM529238(US11198695, Example II-174 | US20240374587, Exampl...)
Affinity DataIC50: 2.16nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704347BDBM704347(US20240374587, Example I'-153 | US12227509, Exampl...)
Affinity DataIC50: 2.23nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704326BDBM704326(US20240374587, Example I'-006 | US12227509, Exampl...)
Affinity DataIC50: 2.25nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528800BDBM528800(US11198695, Example I-8 | US20240374587, Example I...)
Affinity DataIC50: 2.78nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529024BDBM529024(US11198695, Example I-236 | US20240374587, Example...)
Affinity DataIC50: 2.80nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704342BDBM704342(US20240374587, Example I'-142 | US12227509, Exampl...)
Affinity DataIC50: 2.88nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704344BDBM704344(US20240374587, Example I'-145 | US12227509, Exampl...)
Affinity DataIC50: 2.90nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528979BDBM528979(US11198695, Example II-143 | US11198695, Example I...)
Affinity DataIC50: 2.90nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704318BDBM704318(US20240374587, Example II-121)
Affinity DataIC50: 2.91nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704322BDBM704322(US20240374587, Example II-203)
Affinity DataIC50: 2.98nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704343BDBM704343(US20240374587, Example I'-143 | US12227509, Exampl...)
Affinity DataIC50: 3.43nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704345BDBM704345(US20240374587, Example I'-147 | US12227509, Exampl...)
Affinity DataIC50: 3.5nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704315BDBM704315(US20240374587, Example I-276)
Affinity DataIC50: 4.40nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704336BDBM704336(US20240374587, Example I'-130 | US12227509, Exampl...)
Affinity DataIC50: 4.51nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704338BDBM704338(US20240374587, Example I'-136 | US12227509, Exampl...)
Affinity DataIC50: 4.97nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704346BDBM704346(US20240374587, Example I'-151 | US12227509, Exampl...)
Affinity DataIC50: 5.33nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704341BDBM704341(US20240374587, Example I'-141 | US12227509, Exampl...)
Affinity DataIC50: 6.42nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528813BDBM528813(US11198695, Example I-23 | US20240374587, Example ...)
Affinity DataIC50: 6.5nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704334BDBM704334(US20240374587, Example I'-124)
Affinity DataIC50: 6.5nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 529000BDBM529000(US11198695, Example I-212 | US20240374587, Example...)
Affinity DataIC50: 6.90nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704333BDBM704333(US20240374587, Example I'-123 | US12227509, Exampl...)
Affinity DataIC50: 8.48nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704330BDBM704330(US20240374587, Example I'-058 | US12227509, Exampl...)
Affinity DataIC50: 9.78nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704340BDBM704340(US20240374587, Example I'-139 | US12227509, Exampl...)
Affinity DataIC50: 15.8nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 704309BDBM704309(US20240374587, Example I-034)
Affinity DataIC50: 18nMAssay Description:Solutions of the compounds of the present invention in DMSO were each aliquoted into 0.2·μL portions in a 384-well polystyrene microplate produced by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
US Patent