Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 12658
TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718142(US20250042884, Compound I-8)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718139(US20250042884, Compound I-4)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718140(US20250042884, Compound I-5)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718138(US20250042884, Compound I-3)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718136(US20250042884, Compound I-1)
Affinity DataIC50: 3nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718143(US20250042884, Compound I-9)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718144(US20250042884, Compound I-11)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718141(US20250042884, Compound I-6)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718137(US20250042884, Compound I-2)
Affinity DataIC50: 8nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718145(US20250042884, Comparative Compound 2)
Affinity DataIC50: 15.5nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM50136674((R)-duloxetine | LY248685 | (3R)-N-methyl-3-(1-nap...)
Affinity DataIC50: 35.5nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent

TargetHeat shock protein 75 kDa, mitochondrial(Human)
Shanghai Leado Pharmatech Co.

US Patent
LigandPNGBDBM718146(US20250042884, Compound of formula A)
Affinity DataIC50: 75.5nMAssay Description:Ion Works Barracuda (IWB) automated patch clamp detection was used as test method: HEK293 cells stably expressing TRPA1 were placed in DMEM medium co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent