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Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 12795
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729304(((1-(8-methoxyquinazolin-4- yl)azepan-4-yl)methyl)...)
Affinity DataIC50: 10nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729302(((1-(3-cyano-6,7- dimethoxyquinolin-4-yl)azepan-4-...)
Affinity DataIC50: 10nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729289((2-(1-(6,7-dimethoxyquinazolin- 4-yl)azepan-4- yl)...)
Affinity DataIC50: 10nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729290((3-(1-(6,7-dimethoxyquinazolin- 4-yl)azepan-4- yl)...)
Affinity DataIC50: 55nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729283(((1-(6,7-dimethoxyquinazolin-4- yl)azepan-4-yl)met...)
Affinity DataIC50: 55nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729095((R)-((1-(6,7- dimethoxyquinazolin-4-yl)azepan- 4-y...)
Affinity DataIC50: 55nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729305(US20250099493, Compound I-10)
Affinity DataIC50: 100nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729303(((1-(8-methoxyquinolin-4- yl)azepan-4-yl)methyl)ph...)
Affinity DataIC50: 100nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729291(((4-(6,7-dimethoxyquinazolin-4- yl)-1,4-diazepan-1...)
Affinity DataIC50: 100nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 1(Human)
Stingray Therapeutics

US Patent
LigandPNGBDBM729136((S)-((1-(6,7-dimethoxyquinazolin- 4-yl)azepan-4- y...)
Affinity DataIC50: 100nMAssay Description:Materials:Assay Buffer: 1 mM CaCl2), 0.2 mM ZnCl2, 50 mM Tris, pH 9.0. Substrate: 8 mM Thymidine 5′-monophosphate p-nitrophenol ester sodium salt (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent